SCHEMBL13680786

SCHEMBL13680786

O=CCCc1cccc(-c2ccc(OC(F)(F)F)cc2)c1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.46
CHRM1 P11229 1/20 0.46
CHRM3 P20309 1/20 0.46
SLC13A5 Q86YT5 1/20 0.43
TRPV1 Q8NER1 1/20 0.42
SERPINE1 P05121 4/20 0.41
MRGPRX4 Q96LA9 2/20 0.41
ABL1 P00519 1/20 0.41
SCN5A Q14524 1/20 0.40
DAO P14920 1/20 0.40
AGXT P21549 1/20 0.40
MME P08473 1/20 0.39
CHRM5 P08912 2/20 0.39
CA12 O43570 1/20 0.39
CA9 Q16790 1/20 0.39
AURKA O14965 1/20 0.38
TPX2 Q9ULW0 1/20 0.38
ROCK2 O75116 1/20 0.38
ROCK1 Q13464 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5537502 0.84 CHRM2 (0.62) CHRM2CHRM1CHRM3DAOCHRM5
SCHEMBL13680784 0.81 ABL1 (0.50) CHRM2CHRM1CHRM3ABL1
SCHEMBL13680787 0.81 AGXT (0.56) SLC13A5AGXT
SCHEMBL13680798 0.81 CYP1A2 (0.38) CHRM2CHRM1CHRM3SLC13A5MRGPRX4
SCHEMBL8367734 0.81 DRD1 (0.52) MRGPRX4DAOAGXT
SCHEMBL584633 0.80 GPR84 (0.49) CHRM2CHRM1CHRM3TRPV1DAO
SCHEMBL2302446 0.80 FFAR4 (0.46) AGXT
SCHEMBL13099463 0.79 BCL2 (0.51) SLC13A5SERPINE1MRGPRX4ABL1SCN5A
SCHEMBL13680783 0.79 FFAR1 (0.45)
SCHEMBL418611 0.78 GPR52 (0.50) AGXT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed