SCHEMBL13680798

SCHEMBL13680798

O=CCCc1cccc(-c2ccc(OC(F)(F)F)nc2)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
CHRM2 P08172 1/20 0.37
CHRM1 P11229 1/20 0.37
CHRM3 P20309 1/20 0.37
CTSD P07339 1/20 0.36
BACE1 P56817 1/20 0.36
BACE2 Q9Y5Z0 1/20 0.36
HSD17B1 P14061 1/20 0.36
HSD17B2 P37059 1/20 0.36
ELOVL1 Q9BW60 1/20 0.35
ALDH1A1 P00352 1/20 0.34
POLB P06746 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
F2RL3 Q96RI0 3/20 0.34
EGFR P00533 2/20 0.34
FGFR1 P11362 1/20 0.34
GRIN1 Q05586 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680810 0.84 HSD17B1 (0.53) CYP1A2CYP3A4CYP2C9CYP2C19HSD17B1
SCHEMBL13680809 0.81 GRIN1 (0.41) GRIN1GRIN2BMRGPRX4
SCHEMBL13680786 0.81 CHRM2 (0.46) CHRM2CHRM1CHRM3AGXTSLC13A5
SCHEMBL13680797 0.79 CYP11B2 (0.38) GRIN1GRIN2BAGXTCYP4F2CYP4A11
SCHEMBL13680845 0.78 SCN9A (0.41) CYP1A2CYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL13680808 0.77 EPHX2 (0.38) BACE1GRIN1GRIN2BCYP4F2CYP4A11
SCHEMBL13680811 0.73 HIF1A (0.48) CYP1A2CYP3A4HSD17B1HSD17B2ALDH1A1
SCHEMBL13680445 0.73 HSD17B1 (0.46) CTSDBACE1BACE2HSD17B1HSD17B2
SCHEMBL13680787 0.73 AGXT (0.56) AGXTSLC13A5
SCHEMBL13680901 0.73 CYP1A2 (0.36) CYP1A2CYP3A4CYP2C9CYP2C19ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed