SCHEMBL13680797

SCHEMBL13680797

O=CCCc1cccc(-c2ccc(F)nc2)c1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 2/20 0.38
GRIN1 Q05586 3/20 0.36
GRIN2B Q13224 3/20 0.36
CYP2E1 P05181 1/20 0.36
CYP2A6 P11509 1/20 0.36
CYP2B6 P20813 1/20 0.36
CDK8 P49336 2/20 0.36
DRD2 P14416 2/20 0.35
DRD4 P21917 2/20 0.35
DRD3 P35462 2/20 0.35
HIF1A Q16665 1/20 0.35
SRC P12931 1/20 0.35
TAAR1 Q96RJ0 2/20 0.35
DHODH Q02127 1/20 0.34
AGXT P21549 1/20 0.34
CYP4F2 P78329 1/20 0.34
CYP4A11 Q02928 1/20 0.34
CYP11B1 P15538 1/20 0.34
GRM5 P41594 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680808 0.83 EPHX2 (0.38) GRIN1GRIN2BCDK8HIF1ACYP4F2
SCHEMBL13680809 0.82 GRIN1 (0.41) GRIN1GRIN2BCDK8
SCHEMBL5675196 0.81 TAAR1 (0.55) CYP11B2CDK8DRD2TAAR1
SCHEMBL13680810 0.80 HSD17B1 (0.53) CYP2A6
SCHEMBL13680811 0.80 HIF1A (0.48) HIF1ACYP4F2CYP4A11
SCHEMBL13680798 0.79 CYP1A2 (0.38) GRIN1GRIN2BAGXTCYP4F2CYP4A11
SCHEMBL13680805 0.78 EPHX2 (0.55) CYP11B2CYP2E1CYP2A6CYP2B6CYP11B1
SCHEMBL24721758 0.77 BCL2 (0.47) CYP11B2GRIN1GRIN2BCYP2E1CYP2A6
SCHEMBL16675747 0.77 PRKCI (0.53) CYP11B2CYP2E1CYP2A6CYP2B6CDK8
SCHEMBL5215922 0.77 CYP11B2 (0.42) CYP11B2GRIN1GRIN2BCYP2E1CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed