SCHEMBL13680978

SCHEMBL13680978

O=CCCc1ccc(-c2ccc3c(c2)CC(=O)N3)o1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 1/20 0.47
PDE3A Q14432 1/20 0.47
PGR P06401 4/20 0.44
GRIA1 P42261 3/20 0.44
CACNG8 Q8WXS5 3/20 0.44
CYP1A2 P05177 1/20 0.42
CYP11B1 P15538 1/20 0.42
CYP11B2 P19099 1/20 0.42
AHR P35869 2/20 0.41
CDC7 O00311 1/20 0.41
CCNE1 P24864 1/20 0.41
CDK2 P24941 1/20 0.41
DBF4 Q9UBU7 1/20 0.41
PDE4A P27815 1/20 0.39
PDE4B Q07343 1/20 0.39
PDE4C Q08493 1/20 0.39
PDE4D Q08499 1/20 0.39
MAOB P27338 1/20 0.37
BRD4 O60885 2/20 0.37
CREBBP Q92793 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680973 0.90 CRBN (0.42) PDE3BPDE3APGRGRIA1CACNG8
SCHEMBL13680968 0.76 ALDH1A1 (0.35) CYP1A2MAOB
SCHEMBL13680600 0.76 GRIA1 (0.57) PDE3BPDE3APGRGRIA1CACNG8
SCHEMBL16090326 0.76 PGR (0.57) PDE3BPDE3APGRGRIA1CACNG8
SCHEMBL23222381 0.76 HRH1 (0.51) PDE3BPDE3APGRGRIA1CACNG8
SCHEMBL13680969 0.75 GSK3B (0.43)
SCHEMBL13681010 0.75 PDE3B (0.50) PDE3BPDE3APGRGRIA1CACNG8
SCHEMBL13681001 0.74 HSD17B1 (0.44) PGRCYP1A2CYP11B1CYP11B2MAOB
SCHEMBL13680985 0.73 PRF1 (0.52)
SCHEMBL13680976 0.71 MAPT (0.50) PDE3BPDE3AGRIA1CACNG8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed