SCHEMBL13680973

SCHEMBL13680973

O=CCCc1ccc(-c2ccc3c(c2)NC(=O)C3)o1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 3/20 0.42
AHR P35869 3/20 0.41
CMA1 P23946 2/20 0.41
EIF2AK2 P19525 1/20 0.40
S1PR1 P21453 1/20 0.38
KDM1A O60341 1/20 0.37
BRD4 O60885 1/20 0.37
CREBBP Q92793 1/20 0.37
TDP2 O95551 2/20 0.36
PDK2 Q15119 1/20 0.36
PDE3B Q13370 1/20 0.35
PDE3A Q14432 1/20 0.35
ALDH1A1 P00352 4/20 0.34
MAPT P10636 3/20 0.34
PKM P14618 3/20 0.34
KDM4E B2RXH2 2/20 0.34
HPGD P15428 2/20 0.34
HTT P42858 2/20 0.34
HSD17B10 Q99714 2/20 0.34
GFER P55789 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680978 0.90 PDE3B (0.47) AHRBRD4CREBBPTDP2PDK2
SCHEMBL13680598 0.76 CRBN (0.50) CRBNAHRCMA1EIF2AK2S1PR1
SCHEMBL13681000 0.76 CRBN (0.40) CRBNAHRCMA1EIF2AK2S1PR1
SCHEMBL13680968 0.73 ALDH1A1 (0.35) ALDH1A1MAPTPKMKDM4EHPGD
SCHEMBL13680969 0.72 GSK3B (0.43)
SCHEMBL13681001 0.72 HSD17B1 (0.44) ALDH1A1MAPTPKMKDM4EHPGD
SCHEMBL13680976 0.71 MAPT (0.50) PDE3BPDE3AALDH1A1MAPTPKM
SCHEMBL13680985 0.71 PRF1 (0.52) MAPT
SCHEMBL13681029 0.70 ALDH1A1 (0.36) ALDH1A1MAPTPKMKDM4EHPGD
SCHEMBL13680864 0.69 ALDH1A1 (0.63) ALDH1A1MAPTPKMKDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed