SCHEMBL16200054

SCHEMBL16200054

Cn1nc(-c2cccnc2)c(Cl)c1C(F)(F)F

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 3/20 0.45
SMN1; SMN2 Q16637 2/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
RXFP1 Q9HBX9 1/20 0.43
CYP2A6 P11509 4/20 0.42
ALDH1A1 P00352 4/20 0.42
CYP2A13 Q16696 1/20 0.42
PDK2 Q15119 1/20 0.41
CYP2E1 P05181 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2B6 P20813 1/20 0.40
CYP2C19 P33261 1/20 0.40
PTGS1 P23219 2/20 0.39
PTGS2 P35354 2/20 0.39
KDM4E B2RXH2 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14039900 0.83 ALDH1A1 (0.50) SMN1; SMN2ALDH1A1CYP2C9CYP2C19KDM4E
SCHEMBL16200057 0.82 MAPK14 (0.42) NPC1RAB9AALDH1A1CYP2C9CYP2C19
SCHEMBL28851687 0.80 P2RX7 (0.43) P2RX7SMN1; SMN2NPC1RAB9ARXFP1
SCHEMBL16200063 0.79 ALDH1A1 (0.48) P2RX7CYP2A6ALDH1A1CYP2A13CYP2E1
SCHEMBL14039556 0.78 NT5E (0.41) ALDH1A1PTGS2KDM4ECYP1A2CYP3A4
SCHEMBL8108697 0.78 SLC34A1 (0.38) SMN1; SMN2CYP2A6ALDH1A1CYP2C9CYP2C19
SCHEMBL2690242 0.78 CYP2A6 (0.45) P2RX7CYP2A6ALDH1A1CYP2A13CYP2E1
SCHEMBL13683096 0.77 LMNA (0.46) P2RX7SMN1; SMN2NPC1RAB9ARXFP1
SCHEMBL2690686 0.77 CYP2A6 (0.44) P2RX7CYP2A6ALDH1A1CYP2A13CYP2E1
SCHEMBL16200053 0.76 SLC34A1 (0.44) P2RX7SMN1; SMN2RAB9APTGS1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720545-B1 BICYCLIC AND BRIDGED NITROGEN HETEROCYCLES CHEMOCENTRYX INC (US) 2014-10-29 EP disclosed