SCHEMBL16200083

SCHEMBL16200083

Cc1nn(C)c(-c2cccnc2)c1Cl

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.48
CYP11B2 P19099 3/20 0.47
CYP2A6 P11509 7/20 0.44
CYP1A2 P05177 2/20 0.44
CYP3A4 P08684 2/20 0.44
CYP2A13 Q16696 1/20 0.42
P2RX7 Q99572 1/20 0.42
CYP11B1 P15538 1/20 0.42
MAOA P21397 1/20 0.42
LMNA P02545 1/20 0.41
CYP2C9 P11712 2/20 0.41
CYP2C19 P33261 2/20 0.41
CYP2E1 P05181 1/20 0.41
CYP2B6 P20813 1/20 0.41
NPY5R Q15761 1/20 0.40
HSD17B10 Q99714 2/20 0.40
KDM4E B2RXH2 1/20 0.40
HTT P42858 1/20 0.40
HK1 P19367 1/20 0.40
HKDC1 Q2TB90 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30522569 0.83 CYP11B2 (0.53) ALDH1A1CYP11B2CYP2A6CYP1A2CYP3A4
SCHEMBL16200260 0.80 SMN1; SMN2 (0.39) ALDH1A1P2RX7LMNAKDM4E
SCHEMBL13683096 0.79 LMNA (0.46) ALDH1A1CYP11B2CYP2A6CYP1A2CYP3A4
SCHEMBL16200223 0.79 SMN1; SMN2 (0.41) ALDH1A1LMNA
SCHEMBL16200063 0.77 ALDH1A1 (0.48) ALDH1A1CYP11B2CYP2A6CYP1A2CYP3A4
SCHEMBL30522602 0.77 CYP11B2 (0.49) ALDH1A1CYP11B2CYP2A6CYP1A2CYP3A4
SCHEMBL16200236 0.75 LMNA (0.44) ALDH1A1LMNAKDM4E
SCHEMBL16200254 0.75 MEN1 (0.47) ALDH1A1CYP2A6LMNA
SCHEMBL30230959 0.75 CYP11B2 (0.50) ALDH1A1CYP11B2CYP2A6CYP1A2CYP3A4
SCHEMBL16200256 0.74 L3MBTL1 (0.45) ALDH1A1MAOALMNAKDM4EHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720545-B1 BICYCLIC AND BRIDGED NITROGEN HETEROCYCLES CHEMOCENTRYX INC (US) 2014-10-29 EP disclosed