SCHEMBL13711065

SCHEMBL13711065

CNC(C(N)=O)c1ccc(F)c(F)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.44
CES1 P23141 2/20 0.44
APP P05067 1/20 0.42
MME P08473 1/20 0.39
S1PR1 P21453 1/20 0.37
S1PR3 Q99500 1/20 0.37
PDPK1 O15530 1/20 0.37
ROCK2 O75116 2/20 0.36
CHRNA1 P02708 1/20 0.36
CHRNG P07510 1/20 0.36
CHRNB1 P11230 1/20 0.36
CHRNB2 P17787 1/20 0.36
SLC6A2 P23975 1/20 0.36
CHRNB4 P30926 1/20 0.36
CHRNA3 P32297 1/20 0.36
CHRNA4 P43681 1/20 0.36
SLC6A3 Q01959 1/20 0.36
CHRND Q07001 1/20 0.36
AKR1C3 P42330 1/20 0.36
AKR1C2 P52895 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23112517 0.84 MME (0.46) CES2CES1APPMMES1PR1
SCHEMBL13707908 0.83 APP (0.43) CES2CES1APPMMES1PR1
SCHEMBL13710928 0.80 HDAC3 (0.44) ROCK2
SCHEMBL13710925 0.78 HDAC4 (0.50) CES2CES1ROCK2
SCHEMBL23716167 0.77 FFAR2 (0.47) ROCK2SLC6A3
SCHEMBL13710935 0.75 ROCK2 (0.48) ROCK2
SCHEMBL23716154 0.75 ROCK2 (0.48) ROCK2
SCHEMBL19716839 0.74 CES2 (0.62) CES2CES1APPMMEAKR1C3
SCHEMBL15787297 0.74 LMNA (0.47) ROCK2
SCHEMBL20141045 0.74 MEN1 (0.44) PDPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7595299-B2 Peptides as NS3-serine protease inhibitors of hepatitis C virus SCHERING CORPORATION (US) 2009-09-29 US disclosed
US-7169760-B2 Peptides as NS3-serine protease inhibitors of hepatitis C virus SCHERING CORPORATION (US) 2007-01-30 US disclosed