SCHEMBL13730604

SCHEMBL13730604

Cc1ccc(-c2ccnc(N)c2N)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 4/20 0.52
NOS2 P35228 4/20 0.52
MEN1 O00255 4/20 0.42
KMT2A Q03164 4/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
KDR P35968 4/20 0.42
LRRK2 Q5S007 2/20 0.40
MAP4K4 O95819 1/20 0.40
SRC P12931 1/20 0.39
USP7 Q93009 1/20 0.39
KDM4E B2RXH2 2/20 0.38
LMNA P02545 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
MAPT P10636 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
POLB P06746 1/20 0.38
PPARG P37231 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5319523 0.81 NOS2 (0.44) NOS3NOS2NPC1RAB9AKDR
SCHEMBL11901650 0.80 MAP4K4 (0.46) NOS3NOS2NPC1RAB9AKDR
SCHEMBL17555671 0.80 CDK2 (0.43) NOS3NOS2KDRLRRK2MAP4K4
SCHEMBL1823930 0.79 DYRK1A (0.53) NOS3NOS2MEN1KMT2ANPC1
SCHEMBL1165179 0.79 GSK3B (0.47) NOS3NOS2KDRLRRK2MAP4K4
SCHEMBL5973721 0.79 MAPT (0.47) NOS3NOS2MEN1KMT2ANPC1
SCHEMBL11901043 0.78 MAP4K4 (0.48) NOS3NOS2MEN1KMT2ANPC1
Iodide SCHEMBL31385461 0.78 MAPT (0.46) NOS3NOS2MEN1KMT2ANPC1
SCHEMBL4582572 0.76 MKNK1 (0.59) NOS3NOS2MEN1KMT2ANPC1
SCHEMBL3243063 0.76 KIF11 (0.47) NOS3NOS2MAP4K4GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108640872-B GSK-3 inhibitor and preparation method and application thereof 山东大学 2020-04-07 CN disclosed
WO-2012146667-A1 IMIDAZOPYRIDINE DERIVATIVES AS PI3K INHIBITORS ALMIRALL, S.A. (ES) 2012-11-01 WO disclosed