Ethacridine

Ethacridine

SCHEMBL138154

CC(O)C(=O)O.CCOc1ccc2nc3cc(N)ccc3c(N)c2c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

CHRM1DRD2DRD3DRD4HDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HTR2APDE3ASIGMAR1

The experimentally established mechanism targets of Ethacridine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 1.00
KMT2A Q03164 3/20 1.00
CASP7 P55210 3/20 1.00
CASP1 P29466 2/20 1.00
KDM4E B2RXH2 2/20 1.00
ALDH1A1 P00352 2/20 1.00
HPGD P15428 2/20 1.00
HSD17B10 Q99714 2/20 1.00
MAPT P10636 1/20 1.00
MAPK1 P28482 1/20 1.00
BLM P54132 2/20 0.80
TERT O14746 1/20 0.80
ABCB11 O95342 1/20 0.80
LMNA P02545 1/20 0.80
THRB P10828 1/20 0.80
APAF1 O14727 1/20 0.52
POLB P06746 1/20 0.52
CASP3 P42574 1/20 0.52
CASP6 P55212 1/20 0.52
CASP8 Q14790 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ethacridine SCHEMBL30775016 1.00 MEN1 (1.00) MEN1KMT2ACASP7CASP1KDM4E
Ethacridine SCHEMBL30006678 1.00 MEN1 (1.00) MEN1KMT2ACASP7CASP1KDM4E
Ethacridine SCHEMBL31197660 1.00 MEN1 (1.00) MEN1KMT2ACASP7CASP1KDM4E
Ethacridine SCHEMBL8676831 0.99 MEN1 (0.98) MEN1KMT2ACASP7CASP1KDM4E
Ethacridine SCHEMBL1649444 0.99 MEN1 (0.98) MEN1KMT2ACASP7CASP1KDM4E
Ethacridine SCHEMBL29568982 0.99 MEN1 (0.98) MEN1KMT2ACASP7CASP1KDM4E
Ethacridine SCHEMBL29355684 0.99 MEN1 (0.98) MEN1KMT2ACASP7CASP1KDM4E
Ethacridine SCHEMBL3967085 0.98 MEN1 (0.96) MEN1KMT2ACASP7CASP1KDM4E
Lactic Acid SCHEMBL8375854 0.95 MEN1 (0.91) MEN1KMT2ACASP7CASP1KDM4E
Ethacridine SCHEMBL193949 0.89 MEN1 (1.00) MEN1KMT2ACASP7CASP1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1623 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260144911-A1 BURN WOUND TREATMENT Marie's Original Formulas LLC (US) 2026-05-28 US claimed
US-20260144910-A1 BURN WOUND TREATMENT Marie's Original Formulas LLC (US) 2026-05-28 US claimed
EP-4640238-A1 THERAPEUTIC AGENT FOR PULMONARY DISEASE, HEPATIC DISEASE OR RENAL DISEASE, WHICH CONTAINS PGAM-CHK1 BINDING INHIBITOR Kyoto University (JP) 2025-10-29 EP claimed
US-20250213551-A1 WOUND TREATMENT Marie's Original Formulas LLC 2025-07-03 US claimed
US-20250186651-A1 HYDROGEL-BASED TOPICAL WOUND DRESSING CONTAINING PROTEIN EXTRACT T&R BIOFAB CO., LTD. (KR) 2025-06-12 US claimed
US-12311074-B1 Burn wound treatment Marie's Original Formulas LLC (US) 2025-05-27 US claimed
US-12274830-B2 Nitric oxide inhalation therapy for infants with bronchiolitis BEYOND AIR LTD (IL) 2025-04-15 US claimed
US-12247246-B2 Identification of inhibitors of TcpC and TIR NADase activity WASHINGTON UNIVERSITY (US) 2025-03-11 US claimed
CN-119280450-A Medical fabric dressing with long-acting disinfection and sterilization functions and preparation method thereof 孙国明 2025-01-10 CN claimed
US-20250003952-A1 SENOLYTIC DRUG SCREENING METHOD AND SENOLYTIC DRUG KYOTO UNIVERSITY (JP) 2025-01-02 US claimed
EP-0071647-B1 PROCESS FOR RECOVERING INTERFERON GREEN CROSS CORPORATION (JP) 1984-12-05 EP claimed
US-4455146-A THERMOPLASTIC ELASTOMERS, OILS OR FATTY ACID, TACKFIER, AND A MEDICINE HISAMITSU PHARMACEUTICAL CO., LTD. (JP) 1984-06-19 US claimed
EP-0097440-A1 Method and kit for removing and assaying complement system fragments THE UPJOHN COMPANY (US) 1984-01-04 EP claimed
EP-0071647-A1 PROCESS FOR RECOVERING INTERFERON GREEN CROSS CORPORATION (JP) 1983-02-16 EP claimed
US-4137222-A GLOBULINS, PLASMIN, FROM HUMAN BLOOD INSTITUT MERIEUX (FR) 1979-01-30 US claimed
US-4129648-A BLOOD PLASMA OR SERUM EXTRACT COLLIER HARRY O J 1978-12-12 US claimed
US-4104125-A Process for producing human lysozyme THE GREEN CROSS CORPORATION (JP) 1978-08-01 US claimed
US-4017470-A Method for preparing a heat-stable plasma protein solution from paste IV-1 THE GREEN CROSS CORPORATION (JA) 1977-04-12 US claimed
US-3972858-A SILICIC ACID, ELUTION BEHRINGWERKE AKTIENGESELLSCHAFT 1976-08-03 US claimed
US-3946105-A CHROMATOGRAPHY, DIALYSIS, IMMUNIZATION, BLEEDING, ABSORPTION KOWA COMPANY, LTD. (JA) 1976-03-23 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12247246-B2 Identification of inhibitors of TcpC and TIR NADase activity NADK, NAPRT, TIPARP MEN1 3678/4885KMT2A 3095/4885CASP7 4463/4885
US-20260144910-A1 BURN WOUND TREATMENT CUTA, COL1A1, MMP1 MEN1 4599/4885KMT2A 4768/4885CASP7 1204/4885
US-20260144911-A1 BURN WOUND TREATMENT CUTA, LIPG, COL1A1 MEN1 4650/4885KMT2A 4740/4885CASP7 889/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.