SCHEMBL13824871

SCHEMBL13824871

COc1ccc(-c2cccc3cc(C)oc23)c2cc(C)oc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.47
ALDH1A1 P00352 3/20 0.47
SMN1; SMN2 Q16637 3/20 0.47
HPGD P15428 2/20 0.47
HSD17B10 Q99714 2/20 0.47
LMNA P02545 1/20 0.43
RECQL P46063 1/20 0.43
NPC1 O15118 4/20 0.41
RAB9A P51151 4/20 0.41
MAPT P10636 2/20 0.41
PKM P14618 1/20 0.41
CYP3A4 P08684 1/20 0.41
ADORA3 P0DMS8 3/20 0.40
ADORA2A P29274 3/20 0.40
KMT2A Q03164 4/20 0.40
MEN1 O00255 3/20 0.39
CA12 O43570 2/20 0.38
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38
CA9 Q16790 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL73415 0.80 LMNA (0.58) KDM4EALDH1A1SMN1; SMN2HPGDHSD17B10
SCHEMBL13824939 0.70 ALOX5 (0.35)
SCHEMBL20562110 0.70 KDM4E (0.44) KDM4EALDH1A1SMN1; SMN2HPGDHSD17B10
SCHEMBL3705592 0.70 IDO1 (0.47) KDM4EALDH1A1SMN1; SMN2HPGDHSD17B10
SCHEMBL16345751 0.70 F2RL3 (0.46) KDM4EALDH1A1SMN1; SMN2HPGDHSD17B10
SCHEMBL25469348 0.68 KDM4E (0.43) KDM4EALDH1A1SMN1; SMN2HPGDHSD17B10
SCHEMBL28592427 0.68 ALDH1A1 (0.64) KDM4EALDH1A1SMN1; SMN2HPGDHSD17B10
SCHEMBL2128656 0.67 MCL1 (0.60) KDM4EALDH1A1SMN1; SMN2HPGDHSD17B10
SCHEMBL73726 0.67 ALDH1A1 (0.45) KDM4EALDH1A1SMN1; SMN2HPGDHSD17B10
SCHEMBL7917308 0.67 IMPDH2 (0.51) KDM4EALDH1A1SMN1; SMN2HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012150305-A1 NOVEL ANTIFUNGAL 5,6-DIHYDRO-4H-PYRROLO[1,2-a][1,4]BENZO- DIAZEPINES AND 6H-PYRROLO[1,2-a][1,4]BENZODIAZEPINES SUBSTITUTED WITH HETEROCYCLIC DERIVATIVES JANSSEN PHARMACEUTICA NV (BE) 2012-11-08 WO disclosed