SCHEMBL1397443

SCHEMBL1397443

CCCc1ccc2oc(CN(CCc3ccc(Cl)c(Cl)c3)C(=O)c3cc(Cl)cc4cc[nH]c34)cc2c1

nearest known ligand 0.31

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.31
OPRD1 P41143 1/20 0.31
TSHR P16473 1/20 0.31
S1PR1 P21453 2/20 0.31
IKBKB O14920 1/20 0.30
CHUK O15111 1/20 0.30
S1PR3 Q99500 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1397731 0.95 TP53 (0.32) OPRM1OPRD1IKBKBCHUK
SCHEMBL1397655 0.92 MAPT (0.35) TSHRIKBKBCHUK
SCHEMBL1397538 0.89 THRB (0.32) IKBKBCHUK
SCHEMBL1397640 0.89 IKBKB (0.38) OPRM1OPRD1TSHRIKBKBCHUK
SCHEMBL1397802 0.89 MAOB (0.36) IKBKBCHUK
SCHEMBL1397686 0.87 TP53 (0.35) IKBKBCHUK
SCHEMBL1397683 0.85 MAPT (0.33) IKBKBCHUK
SCHEMBL1397462 0.83 CCR2 (0.35)
SCHEMBL1397663 0.77 C5AR1 (0.34) IKBKBCHUK
SCHEMBL1397826 0.76 C5AR1 (0.35) IKBKBCHUK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2007726-B1 BENZAMIDE AND HETEROARENE DERIVATIVES AS CETP INHIBITORS HOFFMANN LA ROCHE (CH) 2011-03-02 EP disclosed