SCHEMBL13985299

SCHEMBL13985299

O=c1cc(CF)nc([C@H]2CC[C@@H](C(F)(F)F)CC2)n1-c1ccc(F)cc1

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 3/20 0.35
TRPA1 O75762 1/20 0.34
GRIA2 P42262 3/20 0.34
GRIN2A Q12879 3/20 0.34
GRIN1 Q05586 2/20 0.34
ALDH1A1 P00352 4/20 0.33
SCN9A Q15858 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
NPC1 O15118 3/20 0.32
RAB9A P51151 3/20 0.32
SMN1; SMN2 Q16637 3/20 0.32
HPGD P15428 2/20 0.32
AOC3 Q16853 1/20 0.32
MAPT P10636 1/20 0.32
LMNA P02545 1/20 0.31
HTT P42858 1/20 0.31
MDM2 Q00987 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4755656 0.84 MEN1 (0.39) MCHR1GRIA2GRIN2AGRIN1ALDH1A1
SCHEMBL4755659 0.84 MEN1 (0.39) MCHR1GRIA2GRIN2AGRIN1ALDH1A1
SCHEMBL4755635 0.81 AVPR1A (0.38) MCHR1MEN1KMT2ASMN1; SMN2MAPT
SCHEMBL4755639 0.81 AVPR1A (0.38) MCHR1MEN1KMT2ASMN1; SMN2MAPT
SCHEMBL13985226 0.81 TBK1 (0.33)
SCHEMBL4755622 0.80 AVPR1A (0.37) MCHR1KMT2ASMN1; SMN2LMNA
SCHEMBL4755627 0.80 AVPR1A (0.37) MCHR1KMT2ASMN1; SMN2LMNA
SCHEMBL13985227 0.78 NOTUM (0.39) SCN9A
SCHEMBL13985415 0.78 AVPR1A (0.36) MCHR1ALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL13985528 0.78 MCHR1 (0.38) MCHR1ALDH1A1MAPTLMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008156607-A1 SUBSTITUTED PYRIMIDINONES NEUROGEN CORPORATION (US) 2008-12-24 WO disclosed