SCHEMBL1404763

SCHEMBL1404763

CC(=O)C=Cc1cccc(Cl)c1O

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IAPP P10997 4/20 0.69
MAPT P10636 5/20 0.58
LMNA P02545 1/20 0.58
KDM4E B2RXH2 2/20 0.49
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
TDP1 Q9NUW8 2/20 0.45
NFKB1 P19838 2/20 0.45
NFKB2 Q00653 2/20 0.45
RELA Q04206 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
POLB P06746 1/20 0.45
ALOX12 P18054 1/20 0.45
HTT P42858 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
HSP90AA1 P07900 1/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC8 Q9BY41 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
GSR P00390 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1404762 1.00 IAPP (0.69) IAPPMAPTLMNAKDM4EMEN1
SCHEMBL1447672 0.83 MAPT (0.63) IAPPMAPTLMNAKDM4EMEN1
SCHEMBL31356685 0.83 MAPT (0.63) IAPPMAPTLMNAKDM4EMEN1
SCHEMBL1447675 0.83 MAPT (0.63) IAPPMAPTLMNAKDM4EMEN1
SCHEMBL7177478 0.81 IAPP (1.00) IAPPMAPTLMNAKDM4ETDP1
SCHEMBL26046362 0.81 IAPP (1.00) IAPPMAPTLMNAKDM4ETDP1
SCHEMBL1404990 0.80 IAPP (0.71) IAPPMAPTLMNAKDM4EMEN1
SCHEMBL1404989 0.80 IAPP (0.71) IAPPMAPTLMNAKDM4EMEN1
SCHEMBL14375297 0.79 IAPP (0.51) IAPPMAPTLMNAKDM4EMEN1
SCHEMBL1405081 0.79 IAPP (0.69) IAPPMAPTLMNAKDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079747-B1 HETEROCYCLIC COMPOUNDS USEFUL AS ANABOLIC AGENTS FOR LIVESTOCK ANIMALS PFIZER LTD (GB) 2011-03-09 EP disclosed
US-20080161288-A1 COMPOUNDS PFIZER INC. 2008-07-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080161288-A1 COMPOUNDS ADRB2, ADRB1, ADRA2C IAPP 1485/4885MAPT 1735/4885LMNA 1543/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.