SCHEMBL14101204

SCHEMBL14101204

CC(C)(C)OC(=O)N1CCc2ccc(C=O)cc2C1

nearest known ligand 0.69

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 2/20 0.69
ESR2 Q92731 2/20 0.63
HDAC1 Q13547 1/20 0.56
MAPK1 P28482 2/20 0.46
MAPT P10636 3/20 0.44
DDB1 Q16531 1/20 0.44
CRBN Q96SW2 1/20 0.44
ABHD6 Q9BV23 3/20 0.44
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
IGF1R P08069 1/20 0.42
ESR1 P03372 1/20 0.41
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
NAMPT P43490 1/20 0.40
GHSR Q92847 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29590724 1.00 NR1H2 (0.69) NR1H2ESR2HDAC1MAPK1MAPT
SCHEMBL2222982 0.95 ESR2 (0.70) NR1H2ESR2HDAC1MAPK1MAPT
SCHEMBL31084557 0.95 ESR2 (0.70) NR1H2ESR2HDAC1MAPK1MAPT
SCHEMBL31281068 0.92 ESR2 (0.59) NR1H2ESR2HDAC1MAPK1MAPT
SCHEMBL12608362 0.92 ESR2 (0.59) NR1H2ESR2HDAC1MAPK1MAPT
SCHEMBL3872976 0.89 HDAC1 (0.67) NR1H2ESR2HDAC1MAPK1DDB1
SCHEMBL30091900 0.89 HDAC1 (0.67) NR1H2ESR2HDAC1MAPK1DDB1
SCHEMBL13538178 0.84 ESR2 (0.69) NR1H2ESR2HDAC1MAPK1MAPT
SCHEMBL3185199 0.83 HDAC1 (0.64) NR1H2ESR2HDAC1MAPK1MAPT
SCHEMBL3178393 0.83 HDAC1 (0.64) NR1H2ESR2HDAC1MAPK1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 35 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12441726-B2 Compounds and uses thereof FOGHORN THERAPEUTICS, INC. (US) 2025-10-14 US disclosed
CN-115297861-B Compounds and uses thereof 福宏治疗公司 2024-07-12 CN disclosed
US-12024531-B2 Immunoproteasome inhibitors PRINCIPIA BIOPHARMA INC. (US) 2024-07-02 US disclosed
US-12024531-B2 Immunoproteasome inhibitors PRINCIPIA BIOPHARMA INC. (US) 2024-07-02 US disclosed
US-12024531-B2 Immunoproteasome inhibitors PRINCIPIA BIOPHARMA INC. (US) 2024-07-02 US disclosed
US-20240174659-A1 COMPOUNDS AND METHODS FOR YAP/TEAD MODULATION AND INDICATIONS THEREFOR Opna Bio SA (CH) 2024-05-30 US disclosed
CN-117956996-A Compounds and methods for YAP/TEAD modulation and indications therefor OPNA 生物公司 2024-04-30 CN disclosed
US-20230257372-A1 NOVEL COMPOUNDS AS HISTONE DEACETYLASE 6 INHIBITOR, AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME CHONG KUN DANG PHARMACEUTICAL CORP. (KR) 2023-08-17 US disclosed
US-20230257372-A1 NOVEL COMPOUNDS AS HISTONE DEACETYLASE 6 INHIBITOR, AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME CHONG KUN DANG PHARMACEUTICAL CORP. (KR) 2023-08-17 US disclosed
US-20230257372-A1 NOVEL COMPOUNDS AS HISTONE DEACETYLASE 6 INHIBITOR, AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME CHONG KUN DANG PHARMACEUTICAL CORP. (KR) 2023-08-17 US disclosed
US-9962388-B2 Pyrrolopyrimidine compounds used as TLR7 agonist CHIA TAI TIANQING PHARMACEUTICAL GROUP CO., LTD. (CN) 2018-05-08 US disclosed
US-20170273983-A1 PYRROLOPYRIMIDINE COMPOUNDS USED AS TLR7 AGONIST CHIA TAI TIANQING PHARMACEUTICAL GROUP CO., LTD. (CN) 2017-09-28 US disclosed
US-20170273983-A1 PYRROLOPYRIMIDINE COMPOUNDS USED AS TLR7 AGONIST CHIA TAI TIANQING PHARMACEUTICAL GROUP CO., LTD. (CN) 2017-09-28 US disclosed
US-20170273983-A1 PYRROLOPYRIMIDINE COMPOUNDS USED AS TLR7 AGONIST CHIA TAI TIANQING PHARMACEUTICAL GROUP CO., LTD. (CN) 2017-09-28 US disclosed
EP-3190113-A1 PYRROLOPYRIMIDINE COMPOUNDS USED AS TLR7 AGONIST Chai Tai Tianqing Pharmaceutical Group Co., Ltd. (CN) 2017-07-12 EP disclosed
EP-3190113-A1 PYRROLOPYRIMIDINE COMPOUNDS USED AS TLR7 AGONIST Chai Tai Tianqing Pharmaceutical Group Co., Ltd. (CN) 2017-07-12 EP disclosed
WO-2016023511-A1 PYRROLOPYRIMIDINE COMPOUNDS USED AS TLR7 AGONIST 正大天晴药业集团股份有限公司 2016-02-18 WO disclosed
EP-1501803-B1 TETRAHYDROPYRANYL CYCLOPENTYL TETRAHYDROISOQUINOLINE MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY MERCK & CO INC (US) 2008-08-13 EP disclosed
US-7166614-B2 Tetrahydropyranyl cyclopentyl tetrahydroisoquinoline modulators of chemokine receptor activity MERCK & CO., INC. (US) 2007-01-23 US disclosed
US-7166614-B2 Tetrahydropyranyl cyclopentyl tetrahydroisoquinoline modulators of chemokine receptor activity MERCK & CO., INC. (US) 2007-01-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240174659-A1 COMPOUNDS AND METHODS FOR YAP/TEAD MODULATION AND INDICATIONS THEREFOR YAP1, YES1, LATS1 NR1H2 89/4885ESR2 723/4885HDAC1 1830/4885
US-20230257372-A1 NOVEL COMPOUNDS AS HISTONE DEACETYLASE 6 INHIBITOR, AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME HDAC6, HDAC1, HDAC3 NR1H2 407/4885ESR2 3660/4885HDAC1 2/4885
US-12441726-B2 Compounds and uses thereof VHL, CLN6, TFEB NR1H2 1847/4885ESR2 1378/4885HDAC1 242/4885
US-12024531-B2 Immunoproteasome inhibitors PSMC2, PSMB7, PSMB2 NR1H2 2436/4885ESR2 2340/4885HDAC1 72/4885
US-20170273983-A1 PYRROLOPYRIMIDINE COMPOUNDS USED AS TLR7 AGONIST TLR7, TLR9, TLR1 NR1H2 528/4885ESR2 3207/4885HDAC1 1632/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.