SCHEMBL14136159

SCHEMBL14136159

O=C1NCC(c2ccccc2)C2(CCN(Cc3ccccc3)CC2)O1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRL1 P41146 2/20 0.47
OPRM1 P35372 1/20 0.47
OPRD1 P41143 1/20 0.47
OPRK1 P41145 1/20 0.47
SIGMAR1 Q99720 8/20 0.47
TMEM97 Q5BJF2 1/20 0.47
PLD2 O14939 1/20 0.46
PLD1 Q13393 1/20 0.46
TSHR P16473 2/20 0.45
LMNA P02545 1/20 0.45
CHRM2 P08172 1/20 0.45
ADRA2A P08913 1/20 0.45
CYP2D6 P10635 1/20 0.45
DRD1 P21728 1/20 0.45
KMT2A Q03164 2/20 0.44
MAPT P10636 1/20 0.44
GRIN2D O15399 2/20 0.44
GRIN3B O60391 2/20 0.44
GRIN1 Q05586 2/20 0.44
GRIN2A Q12879 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13864847 0.84 OPRL1 (0.48) OPRL1OPRM1OPRD1OPRK1SIGMAR1
SCHEMBL1138302 0.79 SLC6A9 (0.58) OPRL1OPRM1OPRD1OPRK1
SCHEMBL4462811 0.78 OPRM1 (0.46) OPRL1OPRM1OPRD1OPRK1SIGMAR1
SCHEMBL6006756 0.78 OPRD1 (0.39) OPRL1OPRM1OPRD1SIGMAR1PLD2
SCHEMBL4558250 0.77 CRBN (0.46) SIGMAR1PLD2PLD1TSHRLMNA
SCHEMBL17113644 0.76 OPRM1 (0.50) OPRL1OPRM1OPRD1OPRK1SIGMAR1
SCHEMBL18075896 0.75 SIGMAR1 (0.48) OPRL1OPRM1OPRD1OPRK1SIGMAR1
SCHEMBL2604320 0.75 TSHR (0.75) OPRL1OPRM1OPRD1OPRK1SIGMAR1
SCHEMBL17101341 0.72 SIGMAR1 (0.45) OPRL1OPRM1OPRD1OPRK1SIGMAR1
SCHEMBL17101331 0.71 TSHR (0.68) OPRL1OPRM1OPRD1OPRK1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1390372-B1 1-OXA-3,9-DIAZA-SPIRO'5,5]UNDECAN-2-ONES DERIVATIVES AND ITS USE AS ANTAGONIST OF THE NEURIKININ RECEPTOR HOFFMANN LA ROCHE (CH) 2008-07-16 EP disclosed