SCHEMBL14148757

SCHEMBL14148757

Nc1sc(-c2ccccc2)nc1-c1ccc(F)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 4/20 0.57
ALOX5 P09917 1/20 0.54
PTGS2 P35354 1/20 0.53
ADORA1 P30542 2/20 0.53
ADORA2A P29274 2/20 0.49
DPP4 P27487 1/20 0.47
APP P05067 1/20 0.45
RARA P10276 1/20 0.43
RARB P10826 1/20 0.43
RARG P13631 1/20 0.43
KDM4E B2RXH2 1/20 0.43
POLB P06746 1/20 0.43
RAB9A P51151 1/20 0.43
CDC7 O00311 1/20 0.42
CCNE1 P24864 1/20 0.42
CDK2 P24941 1/20 0.42
DBF4 Q9UBU7 1/20 0.42
ALDH1A1 P00352 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL543631 0.89 ALDH1A1 (0.50) PTGDR2ADORA1ADORA2ARARARARB
SCHEMBL11652829 0.83 ALOX5 (0.54) PTGDR2ALOX5ADORA1ADORA2ADPP4
SCHEMBL14148598 0.83 KDM4E (0.57) PTGDR2ADORA1ADORA2ADPP4RARA
SCHEMBL14148616 0.83 DPP4 (0.50) PTGDR2ADORA1ADORA2ADPP4CDC7
SCHEMBL11287147 0.81 PTGS2 (0.74) PTGDR2ALOX5PTGS2KDM4EALDH1A1
SCHEMBL544858 0.81 CDC7 (0.61) PTGDR2ADORA1ADORA2AKDM4EPOLB
SCHEMBL14148755 0.80 PTGDR2 (0.60) PTGDR2ALOX5ADORA1ADORA2ADPP4
SCHEMBL14148648 0.80 PTGDR2 (0.60) PTGDR2ALOX5ADORA1ADORA2ADPP4
SCHEMBL14148746 0.78 MAPT (0.51) PTGDR2PTGS2APPKDM4ERAB9A
SCHEMBL29272745 0.77 MYC (0.57) ALOX5ADORA1ADORA2AAPPKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008090382-A1 THIAZOLE AND OXAZOLE DERIVATIVES FOR USE IN THE TREATMENT OF PRION DISEASES, CANCER AND CONDITIONS OF THE CENTRAL NERVOUS SYSTEM AS WELL AS IN THE REGULATION OF STEM CELLS THE UNIVERSITY OF SHEFFIELD (GB) 2008-07-31 WO disclosed