SCHEMBL14200846

SCHEMBL14200846

CCCC(CCC)N(Cc1ccc(C)c(C)c1)C(=O)CC(C)(C)C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 1/20 0.36
TAS1R1 Q7RTX1 1/20 0.36
LMNA P02545 2/20 0.35
HDAC1 Q13547 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
NPC1 O15118 1/20 0.32
HPGD P15428 1/20 0.32
RAB9A P51151 1/20 0.32
ALDH1A1 P00352 1/20 0.32
POLB P06746 1/20 0.32
HSD17B10 Q99714 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
UBE2M P61081 1/20 0.31
DCUN1D1 Q96GG9 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
S1PR1 P21453 1/20 0.31
RIPK1 Q13546 1/20 0.31
KDM4E B2RXH2 1/20 0.31
OPRM1 P35372 1/20 0.31
OPRD1 P41143 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14200894 0.92 NPC1 (0.36) TAS1R3TAS1R1LMNAHDAC1HDAC6
SCHEMBL14200896 0.89 LMNA (0.36) TAS1R3TAS1R1LMNAHDAC1HDAC6
SCHEMBL14200765 0.88 TAS1R3 (0.36) TAS1R3TAS1R1LMNAHDAC1HDAC6
SCHEMBL14229924 0.85 TAS1R3 (0.39) TAS1R3TAS1R1LMNAALDH1A1POLB
SCHEMBL14200932 0.85 HPGD (0.40) TAS1R3TAS1R1LMNANPC1HPGD
SCHEMBL14200859 0.85 PSEN1 (0.39) SMN1; SMN2
SCHEMBL14200864 0.85 RIPK1 (0.48) HPGDRAB9AALDH1A1RIPK1KDM4E
SCHEMBL14200776 0.84 NPC1 (0.35) TAS1R3TAS1R1LMNAHDAC1HDAC6
SCHEMBL14200827 0.83 TRPM8 (0.37) TAS1R3TAS1R1LMNAHDAC1HDAC6
SCHEMBL14200831 0.83 LDHA (0.43) LMNANPC1HPGDRAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7365093-B2 Endothelin antagonists ABBOTT LABORATORIES (US) 2008-04-29 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed