SCHEMBL14200860

SCHEMBL14200860

CCCC(C)N(Cc1cccc(OC)c1)C(=O)CC(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TSPO P30536 1/20 0.42
BCHE P06276 1/20 0.42
ACHE P22303 1/20 0.42
CTSK P43235 1/20 0.41
MEN1 O00255 3/20 0.41
ALDH1A1 P00352 3/20 0.41
KMT2A Q03164 3/20 0.41
ROCK2 O75116 1/20 0.41
MAPT P10636 1/20 0.41
KDM4E B2RXH2 1/20 0.41
LMNA P02545 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
TAS1R3 Q7RTX0 1/20 0.41
TAS1R1 Q7RTX1 1/20 0.41
HSD17B2 P37059 2/20 0.41
MEP1B Q16820 1/20 0.41
PTGES O14684 1/20 0.41
TAAR1 Q96RJ0 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14200833 0.93 EPHX2 (0.45) TSPOBCHEACHECTSKMEN1
SCHEMBL14200838 0.91 ALDH1A1 (0.45) TSPOBCHEACHEMEN1ALDH1A1
SCHEMBL14200895 0.90 TSPO (0.43) TSPOBCHEACHECTSKMEN1
SCHEMBL14229517 0.87 TSPO (0.47) TSPOBCHEACHEMEN1ALDH1A1
SCHEMBL14200862 0.85 CTSK (0.48) TSPOBCHEACHECTSKALDH1A1
SCHEMBL14200947 0.85 MEN1 (0.39) MEN1ALDH1A1KMT2AMAPTLMNA
SCHEMBL14200773 0.85 TSPO (0.44) TSPOBCHEACHEMEN1ALDH1A1
SCHEMBL14200767 0.83 LDHA (0.42) ACHEMEN1ALDH1A1KMT2AMAPT
SCHEMBL14200967 0.81 ALDH1A1 (0.42) MEN1ALDH1A1KMT2AKDM4E
SCHEMBL14229398 0.81 EPHX2 (0.50) TSPOBCHEACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7365093-B2 Endothelin antagonists ABBOTT LABORATORIES (US) 2008-04-29 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed