SCHEMBL14229239

SCHEMBL14229239

CCCC(=O)N(CCC)Cc1ccc(C)c(C)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 3/20 0.44
HDAC6 Q9UBN7 3/20 0.44
HDAC3 O15379 1/20 0.44
HDAC2 Q92769 1/20 0.44
NCOR2 Q9Y618 1/20 0.44
POLB P06746 1/20 0.42
APEX1 P27695 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
TP53 P04637 1/20 0.41
GRIN2D O15399 1/20 0.40
GRIN3B O60391 1/20 0.40
GRIN1 Q05586 1/20 0.40
GRIN2A Q12879 1/20 0.40
GRIN2B Q13224 1/20 0.40
GRIN2C Q14957 1/20 0.40
GRIN3A Q8TCU5 1/20 0.40
HSP90AA1 P07900 1/20 0.38
ALDH1A1 P00352 6/20 0.38
HTT P42858 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14229430 0.91 HDAC6 (0.54) HDAC1HDAC6HDAC3HDAC2NCOR2
SCHEMBL14200898 0.84 HDAC1 (0.40) HDAC1HDAC6HDAC3HDAC2NCOR2
SCHEMBL14229280 0.81 RIPK1 (0.48) HDAC1HDAC6HDAC3HDAC2NCOR2
SCHEMBL14229892 0.81 ALDH1A1 (0.47) HDAC1HDAC6HDAC3HDAC2NCOR2
SCHEMBL14228983 0.81 GRIN2D (0.49) POLBAPEX1TDP1TP53GRIN2D
SCHEMBL14229047 0.78 APP (0.50) TP53ALDH1A1HTTKMT2AHPGD
SCHEMBL14228970 0.78 SMN1; SMN2 (0.37) POLBTP53ALDH1A1KMT2ALMNA
SCHEMBL14229924 0.77 TAS1R3 (0.39) POLBTP53ALDH1A1KMT2ALMNA
SCHEMBL14228962 0.77 TRPM8 (0.39) POLBALDH1A1KMT2ALMNALTB4R2
SCHEMBL14200780 0.76 HDAC6 (0.48) HDAC1HDAC6HDAC3HDAC2NCOR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7365093-B2 Endothelin antagonists ABBOTT LABORATORIES (US) 2008-04-29 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed