SCHEMBL14283239

SCHEMBL14283239

CNc1ccc(S(=O)(=O)N2CCCC2)cc1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.70
USP2 O75604 1/20 0.68
HSD17B10 Q99714 1/20 0.62
PKM P14618 2/20 0.59
MEN1 O00255 2/20 0.59
KMT2A Q03164 2/20 0.59
TSHR P16473 1/20 0.59
TDP1 Q9NUW8 1/20 0.59
POLB P06746 3/20 0.58
HTT P42858 3/20 0.58
MAPT P10636 3/20 0.57
SMN1; SMN2 Q16637 2/20 0.57
LMNA P02545 2/20 0.57
NPC1 O15118 1/20 0.57
RAB9A P51151 1/20 0.57
GAA P10253 1/20 0.57
KDM4E B2RXH2 1/20 0.56
TP53 P04637 1/20 0.56
ALOX15 P16050 1/20 0.56
RECQL P46063 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4655484 0.98 USP2 (0.71) ALDH1A1USP2HSD17B10MEN1KMT2A
SCHEMBL13982817 0.96 ALDH1A1 (0.65) ALDH1A1USP2HSD17B10PKMMEN1
SCHEMBL14094061 0.84 L3MBTL1 (0.68) ALDH1A1HSD17B10MEN1KMT2APOLB
SCHEMBL16809210 0.84 MAPT (0.63) ALDH1A1USP2PKMMAPT
SCHEMBL14057770 0.82 KMT2A (0.51) ALDH1A1MEN1KMT2ATDP1HTT
SCHEMBL12455096 0.81 USP2 (0.68) ALDH1A1USP2HSD17B10PKMMEN1
SCHEMBL13982806 0.81 USP2 (0.67) ALDH1A1USP2HSD17B10MEN1KMT2A
SCHEMBL14538786 0.80 AKR1C3 (0.58) ALDH1A1USP2MEN1KMT2ATDP1
SCHEMBL6945990 0.80 USP2 (0.71) ALDH1A1USP2HSD17B10MEN1KMT2A
SCHEMBL12793711 0.80 USP2 (0.71) ALDH1A1USP2HSD17B10PKMMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8975399-B2 Benzenesulfon amide-compound treatment of a pathological condition linked to an excessive effect of TNF VAX-CONSULTING (FR) 2015-03-10 US disclosed
US-8975399-B2 Benzenesulfon amide-compound treatment of a pathological condition linked to an excessive effect of TNF VAX-CONSULTING (FR) 2015-03-10 US disclosed
US-20130123266-A1 TREATMENT OF A PATHOLOGY LINKED TO AN EXCESSIVE EFFECT OF TNF WITH A BENZENE SULPHONAMIDE COMPOUND VAX-CONSULTING (FR) 2013-05-16 US disclosed
US-20130123266-A1 TREATMENT OF A PATHOLOGY LINKED TO AN EXCESSIVE EFFECT OF TNF WITH A BENZENE SULPHONAMIDE COMPOUND VAX-CONSULTING (FR) 2013-05-16 US disclosed
US-20080015183-A1 SUBSTITUTED QUINAZOLIN-4-YLAMINE ANALOGUES NEUROGEN CORPORATION (US) 2008-01-17 US disclosed
US-7304059-B2 Substituted quinazolin-4-ylamine analogues NEUROGEN CORPORATION (US) 2007-12-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080015183-A1 SUBSTITUTED QUINAZOLIN-4-YLAMINE ANALOGUES PIGS, HRH4, GPR88 ALDH1A1 2125/4885USP2 3877/4885HSD17B10 4462/4885
US-20130123266-A1 TREATMENT OF A PATHOLOGY LINKED TO AN EXCESSIVE EFFECT OF TNF WITH A BENZENE SULPHONAMIDE COMPOUND TNF, TNFRSF1A, TRAF6 ALDH1A1 205/4885USP2 1074/4885HSD17B10 1595/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.