SCHEMBL1442829

SCHEMBL1442829

O=S(=O)(O)CC(O)CNC1CCCCC1.[NaH]

nearest known ligand 0.63

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.63
SMN1; SMN2 Q16637 2/20 0.51
HTT P42858 2/20 0.51
ANPEP P15144 2/20 0.44
ERAP2 Q6P179 2/20 0.44
SLC2A1 P11166 1/20 0.41
KMT2A Q03164 4/20 0.37
MEN1 O00255 3/20 0.37
LMNA P02545 3/20 0.37
POLB P06746 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
ADRB2 P07550 1/20 0.36
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5447671 0.98 KDM4E (0.66) KDM4ESMN1; SMN2HTTANPEPERAP2
SCHEMBL2142228 0.98 KDM4E (0.66) KDM4ESMN1; SMN2HTTANPEPERAP2
SCHEMBL157010 0.98 KDM4E (0.66) KDM4ESMN1; SMN2HTTANPEPERAP2
SCHEMBL30287648 0.97 KDM4E (0.63) KDM4ESMN1; SMN2HTTANPEPERAP2
Bicarbonate SCHEMBL23462324 0.93 KDM4E (0.59) KDM4ESMN1; SMN2HTTANPEPERAP2
Hexamethonium SCHEMBL8821557 0.84 KDM4E (0.49) KDM4ESMN1; SMN2HTTANPEPERAP2
SCHEMBL18577849 0.82 KDM4E (0.46) KDM4ESMN1; SMN2HTTANPEPERAP2
SCHEMBL29710685 0.81 KDM4E (0.61) KDM4ESMN1; SMN2HTTANPEPERAP2
Potassium Ion SCHEMBL30898940 0.81 KDM4E (0.61) KDM4ESMN1; SMN2HTTANPEPERAP2
SCHEMBL13359411 0.81 KDM4E (0.43) KDM4ESMN1; SMN2HTTKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 23 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114752035-A High-solid-content aqueous polyurethane dispersion and preparation method and application thereof 浙江大学衢州研究院 2022-07-15 CN claimed
EP-4347928-A1 ELECTROCHEMICAL METAL DEPOSITION SYSTEM AND METHOD NTH Cycle, Inc. (US) 2024-04-10 EP disclosed
US-20240000084-A1 ANTIPATHOGENIC AGENT, ANTIBACTERIAL AGENT, ANTIVIRAL AGENT, PATHOGEN DISPOSAL DEVICE, ANTIPATHOGENIC AGENT PRODUCTION METHOD, ANTIBACTERIAL TREATMENT METHOD, VIRUS INACTIVATION METHOD, AND PATHOGEN DISPOSAL METHOD ACENET INC. (JP) 2024-01-04 US disclosed
WO-2023190598-A1 COMPOSITION アース製薬株式会社 2023-10-05 WO disclosed
US-20230263710-A1 ORAL CARE AGENT OSAKA UNIVERSITY (JP) 2023-08-24 US disclosed
EP-4230042-A1 ANTIPATHOGENIC DRUG, ANTIBACTERIAL AGENT, ANTIVIRAL AGENT, PATHOGEN PROCESSING DEVICE, METHOD FOR PRODUCING ANTIPATHOGENIC DRUG, ANTIBACTERIAL METHOD, VIRUS INACTIVATION METHOD, AND PATHOGEN PROCESSING METHOD Acenet Inc. (JP) 2023-08-23 EP disclosed
US-20230181628-A1 EPITHELIAL CANCER THERAPEUTIC AGENT OSAKA UNIVERSITY (JP) 2023-06-15 US disclosed
EP-4147703-A1 EPITHELIAL CANCER THERAPEUTIC AGENT OSAKA UNIVERSITY (JP) 2023-03-15 EP disclosed
CN-115666593-A Therapeutic agent for epithelial cancer 国立大学法人大阪大学 2023-01-31 CN disclosed
US-20220389601-A1 ELECTROCHEMICAL METAL DEPOSITION SYSTEM AND METHOD Nth Cycle, Inc. (US) 2022-12-08 US disclosed
US-11041097-B2 Polishing composition and method of fabricating semiconductor device using the same SAMSUNG ELECTRONICS CO., LTD. (KR) 2021-06-22 US disclosed
WO-2021066080-A1 DRUG, DRUG MANUFACTURING METHOD, AND WATER PURIFICATION METHOD 株式会社エースネット 2021-04-08 WO disclosed
US-20200255689-A1 POLISHING COMPOSITION AND METHOD OF FABRICATING SEMICONDUCTOR DEVICE USING THE SAME SAMSUNG ELECTRONICS CO., LTD. (KR) 2020-08-13 US disclosed
US-20200171118-A1 RADICAL GENERATING CATALYST, METHOD FOR PRODUCING RADICAL, METHOD FOR PRODUCING OXIDATION REACTION PRODUCT, DRUG, AND DRUG FOR USE IN AGRICULTURE AND LIVESTOCK INDUSTRY ACENET INC. (JP) 2020-06-04 US disclosed
EP-3626339-A1 RADICAL-GENERATING CATALYST, RADICAL PRODUCTION METHOD, OXIDATION REACTION PRODUCT PRODUCTION METHOD, CHEMICAL AGENT, AND CHEMICAL AGENT FOR AGRICULTURE AND LIVESTOCK Acenet Inc. (JP) 2020-03-25 EP disclosed
EP-2475778-B1 Methods and kit for protease enzyme assays 3M INNOVATIVE PROPERTIES CO (US) 2014-10-22 EP disclosed
US-8349580-B2 Methods and kit for protease enzyme assays 3M INNOVATIVE PROPERTIES COMPANY (US) 2013-01-08 US disclosed
EP-2475778-A1 METHODS AND KIT FOR PROTEASE ENZYME ASSAYS 3M Innovative Properties Company (US) 2012-07-18 EP disclosed
US-20120164675-A1 METHODS AND KIT FOR PROTEASE ENZYME ASSAYS 3M INNOVATIVE PROPERTIES COMPANY 2012-06-28 US disclosed
WO-2011031573-A1 METHODS AND KIT FOR PROTEASE ENZYME ASSAYS 3M INNOVATIVE PROPERTIES COMPANY (US) 2011-03-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230263710-A1 ORAL CARE AGENT TAS2R39, TAS2R40, TAS2R45 KDM4E 1296/4885SMN1; SMN2 3710/4885HTT 2471/4885
US-20200171118-A1 RADICAL GENERATING CATALYST, METHOD FOR PRODUCING RADICAL, METHOD FOR PRODUCING OXIDATION REACTION PRODUCT, DRUG, AND DRUG FOR USE IN AGRICULTURE AND LIVESTOCK INDUSTRY PRDX2, PRDX1, PRDX5 KDM4E 1991/4885SMN1; SMN2 4603/4885HTT 3756/4885
US-20230181628-A1 EPITHELIAL CANCER THERAPEUTIC AGENT EPCAM, EGFR, MUC1 KDM4E 3793/4885SMN1; SMN2 4559/4885HTT 4651/4885
US-20240000084-A1 ANTIPATHOGENIC AGENT, ANTIBACTERIAL AGENT, ANTIVIRAL AGENT, PATHOGEN DISPOSAL DEVICE, ANTIPATHOGENIC AGENT PRODUCTION METHOD, ANTIBACTERIAL TREATMENT METHOD, VIRUS INACTIVATION METHOD, AND PATHOGEN DISPOSAL METHOD EIF2AK2, HAO2, ZC3HAV1 KDM4E 4109/4885SMN1; SMN2 3556/4885HTT 94/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.