SCHEMBL144307

SCHEMBL144307

CCS(=O)(=O)Nc1cc(-n2nnn(CCCF)c2=O)c(F)cc1Cl

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 1/20 0.34
PPOX P50336 1/20 0.34
PSIP1 O75475 1/20 0.33
BRAF P15056 5/20 0.32
KCNH2 Q12809 1/20 0.31
AR P10275 1/20 0.31
PGR P06401 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29367340 1.00 EGLN1 (0.34) EGLN1PPOXPSIP1BRAFKCNH2
SCHEMBL10521129 0.87 CA2 (0.35) PPOX
SCHEMBL10519375 0.86 CA2 (0.34) PPOX
Potassium SCHEMBL10519386 0.86 CA2 (0.34) PPOX
SCHEMBL10521007 0.83
SCHEMBL4364051 0.81 BRAF (0.31) BRAF
SCHEMBL9730340 0.81 BRPF1 (0.38) ARPGR
SCHEMBL21381465 0.81 PGR (0.40) ARPGR
SCHEMBL868158 0.80 BRAF (0.41) PSIP1BRAFKCNH2
SCHEMBL9730432 0.79 BRD9 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1889 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3599857-B1 HERBICIDAL MIXTURES BAYER AG (DE) 2023-08-23 EP claimed
CN-110461158-B Herbicidal mixtures comprising 2- [ (2, 4-dichlorophenyl) methyl ] -4, 4-dimethyl-3-isoxazolidone, topramezone and mefenpyr 拜耳公司 2021-12-10 CN claimed
CN-110461157-B Herbicidal mixtures 拜耳公司 2021-11-02 CN claimed
US-20210289781-A1 HERBICIDAL MIXTURES BAYER AKTIENGESELLSCHAFT (DE) 2021-09-23 US claimed
EP-3823450-A1 HERBICIDAL MIXTURES CONTAINING ACLONIFEN AND CINMETHYLIN Bayer Aktiengesellschaft (DE) 2021-05-26 EP claimed
US-20210137117-A1 HERBICIDAL MIXTURES FMC CORPORATION 2021-05-13 US claimed
CN-112469277-A Herbicidal mixtures comprising aclonifen and cinmethylin 拜耳公司 2021-03-09 CN claimed
US-10932467-B2 Herbicidal mixtures BAYER AKTIENGESELLSCHAFT (DE) 2021-03-02 US claimed
EP-3599856-A1 HERBICIDAL MIXTURES CONTAINING 2-[2,4-DICHLOROPHENYL)METHYL]4,4-DIMETHYL-3-ISOXAZOLIDINONE, PYROXASULFONE AND MEFENPYR-DIETHYL Bayer Aktiengesellschaft (DE) 2020-02-05 EP claimed
EP-3599857-A1 HERBICIDAL MIXTURES Bayer Aktiengesellschaft (DE) 2020-02-05 EP claimed
WO-2020016134-A1 HERBICIDAL MIXTURES CONTAINING ACLONIFEN AND CINMETHYLIN BAYER AKTIENGESELLSCHAFT (DE) 2020-01-23 WO claimed
WO-2018172325-A1 HERBICIDAL MIXTURES CONTAINING 2-[2,4-DICHLOROPHENYL)METHYL]4,4-DIMETHYL-3-ISOXAZOLIDINONE, PYROXASULFONE AND MEFENPYR-DIETHYL BAYER AKTIENGESELLSCHAFT (DE) 2018-09-27 WO claimed
US-20140310835-A1 SOYBEAN EVENT SYHT04R AND COMPOSITIONS AND METHODS FOR DETECTION THEREOF SYNGENTA PARTICIPATIONS AG (CH) 2014-10-16 US claimed
US-20140208463-A1 ACTIVE COMPOUND COMBINATIONS COMPRISING SPECIFIC TETRAMIC ACID DERIVATIVES BAYER INTELLECTUAL PROPERTY GMBH (DE) 2014-07-24 US claimed
WO-2013020985-A1 ACTIVE COMPOUND COMBINATIONS COMPRISING SPECIFIC TETRAMIC ACID DERIVATIVES BAYER INTELLECTUAL PROPERTY GMBH (DE) 2013-02-14 WO claimed
WO-2012082542-A2 SOYBEAN EVENT SYHT04R AND COMPOSITIONS AND METHODS FOR DETECTION THEREOF SYNGENTA PARTICIPATIONS AG (CH) 2012-06-21 WO claimed
US-20260144250-A1 SOLVENT-FREE FORMULATIONS OF LOW-MELTING ACTIVE INGREDIENTS BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2026-05-28 US disclosed
US-20260144252-A1 BROMINE- OR IODINE-PARA-SUBSTITUTED [(1,5-DIPHENYL-1H-1,2,4-TRIAZOL-3-YL)OXY]ACETIC ACID DERIVATIVES AND THEIR SALTS, AGENTS FOR PROTECTING USEFUL PLANTS OR CROP PLANTS COMPRISING THEM, METHODS FOR PRODUCING THEM AND THEIR USE AS SAFENERS BAYER AKTIENGESELLSCHAFT (DE) 2026-05-28 US disclosed
EP-0252982-A1 HERBICIDAL 1-ARYL-4-SUSTITUTTED-1,4-DIHYDRO-5H-TETRAZOL-5-ONES AND SULFUR ANALOGS THEREOF FMC Corporation (US) 1988-01-20 EP disclosed
WO-1987003873-A1 HERBICIDAL 1-ARYL-4-SUBSTITUTED-1,4-DIHYDRO-5H-TETRAZOL-5-ONES AND SULFUR ANALOGS THEREOF FMC CORPORATION (US) 1987-07-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260144250-A1 SOLVENT-FREE FORMULATIONS OF LOW-MELTING ACTIVE INGREDIENTS FOXM1, CSDE1, RCC1 EGLN1 2217/4885PPOX 3277/4885PSIP1 66/4885
US-20210289781-A1 HERBICIDAL MIXTURES ATL3, DDT, CLSPN EGLN1 590/4885PPOX 2194/4885PSIP1 2795/4885
US-20260144252-A1 BROMINE- OR IODINE-PARA-SUBSTITUTED [(1,5-DIPHENYL-1H-1,2,4-TRIAZOL-3-YL)OXY]ACETIC ACID DERIVATIVES AND THEIR SALTS, AGENTS FOR PROTECTING USEFUL PLANTS OR CROP PLANTS COMPRISING THEM, METHODS FOR PRODUCING THEM AND THEIR USE AS SAFENERS CBR3, CBR1, CA3 EGLN1 909/4885PPOX 764/4885PSIP1 1672/4885
US-10932467-B2 Herbicidal mixtures DDT, PRDX5, DHX35 EGLN1 194/4885PPOX 912/4885PSIP1 1048/4885
US-20210137117-A1 HERBICIDAL MIXTURES DDT, MTX2, ATL3 EGLN1 274/4885PPOX 1334/4885PSIP1 1852/4885
US-20140208463-A1 ACTIVE COMPOUND COMBINATIONS COMPRISING SPECIFIC TETRAMIC ACID DERIVATIVES DDT, TBCA, CA3 EGLN1 2398/4885PPOX 1245/4885PSIP1 4164/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.