SCHEMBL1443992

SCHEMBL1443992

OCc1cccc(-c2ccc(F)cc2)c1-c1ccc(F)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 3/20 0.43
CD274 Q9NZQ7 3/20 0.43
ENPP1 P22413 1/20 0.43
PDK2 Q15119 2/20 0.42
PRKAA2 P54646 1/20 0.39
PTGS1 P23219 3/20 0.38
SLC6A4 P31645 1/20 0.38
SLC6A3 Q01959 1/20 0.38
PTGS2 P35354 3/20 0.37
NR4A2 P43354 2/20 0.37
FFAR1 O14842 1/20 0.37
FFAR4 Q5NUL3 1/20 0.37
GCGR P47871 2/20 0.36
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
DAPK3 O43293 1/20 0.36
PRKD3 O94806 1/20 0.36
MAP4K4 O95819 1/20 0.36
PAK4 O96013 1/20 0.36
ABL1 P00519 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9720787 0.90 ESR2 (0.42) PDCD1CD274ENPP1PDK2MAP4K4
SCHEMBL9720784 0.88 ESR2 (0.43) PDCD1CD274ENPP1PDK2GCGR
SCHEMBL9720758 0.88 PDCD1 (0.41) PDCD1CD274ENPP1PDK2PRKAA2
SCHEMBL9720754 0.86 PDCD1 (0.42) PDCD1CD274ENPP1PDK2PRKAA2
SCHEMBL27555128 0.85 TTR (0.43) PDCD1CD274ENPP1PDK2PRKAA2
SCHEMBL1443909 0.83 ENPP1 (0.39) ENPP1PTGS1SLC6A4SLC6A3PTGS2
SCHEMBL11494835 0.82 MMP3 (0.49) PDCD1CD274PDK2ABL1
SCHEMBL13824010 0.82 NR4A2 (0.48) PDCD1CD274ENPP1PDK2PTGS1
SCHEMBL1041243 0.82 PDK2 (0.49) PDCD1CD274PDK2PTGS1SLC6A4
SCHEMBL7204765 0.82 PDCD1 (0.62) PDCD1CD274ENPP1PDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12286389-B2 Crystalline form a of 2, 2-bis(4-fluorophenyl)-2-phenylacetamide and preparation method therefor and application thereof Shenzhen Jingtai Technology Co., Ltd (CN) 2025-04-29 US disclosed
US-20220033347-A1 CRYSTALLINE FORM A OF 2, 2-BIS(4-FLUOROPHENYL)-2-PHENYLACETAMIDE AND PREPARATION METHOD THEREFOR AND APPLICATION THEREOF Shenzhen Jingtai Technology Co., Ltd (CN) 2022-02-03 US disclosed
WO-2011034860-A1 TREATMENT METHODS USING TRIARYL METHANE COMPOUNDS ICAGEN, INC. (US) 2011-03-24 WO disclosed
US-20100056637-A1 TREATMENT METHODS USING TRIARYL METHANE COMPOUNDS ICAGEN, INC. (US) 2010-03-04 US disclosed
US-20090036538-A1 TREATMENT METHODS USING TRIARYL METHANE COMPOUNDS ICAGEN, INC. (US) 2009-02-05 US disclosed
EP-1968563-A2 TREATMENT METHODS USING TRIARYL METHANE COMPOUNDS Icagen, Inc. (US) 2008-09-17 EP disclosed
EP-1158971-B1 GARDOS CHANNEL ANTAGONISTS ICAGEN INC (US) 2007-08-22 EP disclosed
US-20070185209-A1 Treatment methods using triaryl methane compounds ICAGEN, INC. (US) 2007-08-09 US disclosed
WO-2007075849-A2 TREATMENT METHODS USING TRIARYL METHANE COMPOUNDS ICAGEN, INC. (US) 2007-07-05 WO disclosed
EP-1158971-A4 GARDOS CHANNEL ANTAGONISTS ICAGEN INC (US) 2003-04-16 EP disclosed
EP-1158971-A1 GARDOS CHANNEL ANTAGONISTS Icagen, Inc. (US) 2001-12-05 EP disclosed
US-6288122-B1 A TRIPHENYL ACETAMIDE ICAGEN, INC. 2001-09-11 US disclosed
WO-2000050026-A1 GARDOS CHANNEL ANTAGONISTS ICAGEN, INC. (US) 2000-08-31 WO disclosed
US-5149707-A 1-((2-FLUOROPHENYL)(4-FLUOROPHENYL)PHENYLMETHYL)-1H-IMIDAZOLE USEFUL AS ANTIFUNGAL AGENT J. URIACH & CIA, S.A. (ES) 1992-09-22 US disclosed
EP-0352352-B1 1-[(2-Fluorophenyl)(4-fluorophenyl)phenylmethyl]-1H-imidazole J. URIACH & CIA. S.A. (ES) 1991-10-16 EP disclosed
EP-0352352-A1 1-[(2-Fluorophenyl)(4-fluorophenyl)phenylmethyl]-1H-imidazole J. URIACH & CIA. S.A. (ES) 1990-01-31 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070185209-A1 Treatment methods using triaryl methane compounds KCNH3, KCNH2, KCNJ2 PDCD1 2723/4885CD274 3480/4885ENPP1 3912/4885
US-20090036538-A1 TREATMENT METHODS USING TRIARYL METHANE COMPOUNDS KCNH3, KCNH2, KCNJ2 PDCD1 2723/4885CD274 3480/4885ENPP1 3912/4885
US-12286389-B2 Crystalline form a of 2, 2-bis(4-fluorophenyl)-2-phenylacetamide and preparation method therefor and application thereof WEE2, WEE1, WASF2 PDCD1 2854/4885CD274 3704/4885ENPP1 3934/4885
US-20220033347-A1 CRYSTALLINE FORM A OF 2, 2-BIS(4-FLUOROPHENYL)-2-PHENYLACETAMIDE AND PREPARATION METHOD THEREFOR AND APPLICATION THEREOF WEE2, WEE1, WASF2 PDCD1 2854/4885CD274 3704/4885ENPP1 3934/4885
US-20100056637-A1 TREATMENT METHODS USING TRIARYL METHANE COMPOUNDS LTC4S, LTB4R2, CYSLTR2 PDCD1 4522/4885CD274 4658/4885ENPP1 2447/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.