Thiobarbituric

Thiobarbituric

SCHEMBL144675

NC(N)=S.O=C1CC(=O)NC(=S)N1

nearest known ligand 0.42

Full drug profile on Sugi Atlas →

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.33
ITGB1 P05556 1/20 0.33
ITGAV P06756 1/20 0.33
ITGA4 P13612 1/20 0.33
ALDH1A1 P00352 1/20 0.32
CYP1A2 P05177 1/20 0.32
HPGD P15428 1/20 0.32
HIF1A Q16665 1/20 0.32
HSD17B10 Q99714 1/20 0.32
GSK3A P49840 1/20 0.31
GSK3B P49841 1/20 0.31
MAPT P10636 1/20 0.30
TSHR P16473 1/20 0.30
ATM Q13315 1/20 0.30
ATR Q13535 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Thiobarbituric SCHEMBL2455746 0.88 ITGB3 (0.32) ITGB3ITGB1ITGAVITGA4ALDH1A1
Thiobarbituric SCHEMBL16027 0.87
Thiobarbituric SCHEMBL31059040 0.87 GSK3A (0.38) ITGB3ITGB1ITGAVITGA4ALDH1A1
Thiobarbituric SCHEMBL8216351 0.84 GSK3A (0.36) ITGB3ITGB1ITGAVITGA4ALDH1A1
Thiobarbituric SCHEMBL2351184 0.84 GSK3A (0.36) ITGB3ITGB1ITGAVITGA4ALDH1A1
Thiobarbituric SCHEMBL2344775 0.84 GSK3A (0.36) ITGB3ITGB1ITGAVITGA4ALDH1A1
Barbituric Acid SCHEMBL28237381 0.82 ALDH1A1 (0.48) ITGB3ITGB1ITGAVITGA4ALDH1A1
Barbituric Acid SCHEMBL4726594 0.79 ALDH1A1 (0.44) ITGB3ITGB1ITGAVITGA4ALDH1A1
Thiobarbituric SCHEMBL7714190 0.75 ALDH1A1 (0.42) ALDH1A1CYP1A2HPGDGSK3AGSK3B
SCHEMBL8028070 0.74

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120059163-A1 Non-linear opticaly active molecules, their synthesis, and use OPTIMER PHOTONICS, INC. (US) 2012-03-08 US disclosed
US-20080004415-A1 Non-linear optically active molecules, their synthesis, and use OPTIMER PHOTONICS, INC. (US) 2008-01-03 US disclosed
EP-1742906-A2 NON-LINEAR OPTICALLY ACTIVE MOLECULES, THEIR SYNTHESIS, AND USE Optimer Photonics, Inc. (US) 2007-01-17 EP disclosed
WO-2005119315-A2 NON-LINEAR OPTICALLY ACTIVE MOLECULES, THEIR SYNTHESIS, AND USE OPTIMER PHOTONICS, INC. (US) 2005-12-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120059163-A1 Non-linear opticaly active molecules, their synthesis, and use INCENP, CYBA, ADCY5 ITGB3 1468/4885ITGB1 2163/4885ITGAV 3775/4885
US-20080004415-A1 Non-linear optically active molecules, their synthesis, and use INCENP, CYBA, PAICS ITGB3 1795/4885ITGB1 2735/4885ITGAV 3811/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.