SCHEMBL144993

SCHEMBL144993

COc1ccc2nc(Cl)sc2c1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.69
CYP1A2 P05177 2/20 0.65
CYP3A4 P08684 2/20 0.65
CYP2C19 P33261 2/20 0.65
PDK1 Q15118 1/20 0.63
MAPT P10636 4/20 0.56
NPC1 O15118 4/20 0.56
RAB9A P51151 4/20 0.56
SMN1; SMN2 Q16637 4/20 0.56
MEN1 O00255 3/20 0.56
TSHR P16473 1/20 0.56
APP P05067 4/20 0.55
HTT P42858 2/20 0.54
DYRK1A Q13627 1/20 0.54
NFKB1 P19838 1/20 0.54
NFKB2 Q00653 1/20 0.54
RELA Q04206 1/20 0.54
GAA P10253 2/20 0.52
GLA P06280 1/20 0.52
ALDH1A1 P00352 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL779852 0.86 NPC1 (0.54) KMT2ACYP1A2CYP3A4CYP2C19PDK1
SCHEMBL778394 0.81 KMT2A (0.63) KMT2ACYP1A2CYP3A4CYP2C19PDK1
SCHEMBL1748243 0.81 KMT2A (1.00) KMT2ACYP1A2CYP3A4CYP2C19MAPT
SCHEMBL27917560 0.81 APP (0.74) NPC1RAB9ASMN1; SMN2APPGAA
SCHEMBL299010 0.80 CYP1A2 (0.67) KMT2ACYP1A2CYP3A4CYP2C19PDK1
SCHEMBL422166 0.80 CYP1A2 (0.67) KMT2ACYP1A2CYP3A4CYP2C19PDK1
SCHEMBL10531693 0.79 CA2 (0.63) KMT2ACYP1A2CYP3A4CYP2C19NPC1
SCHEMBL30189879 0.79 KMT2A (0.60) KMT2ACYP1A2CYP3A4CYP2C19PDK1
SCHEMBL1748095 0.79 KMT2A (0.78) KMT2ACYP1A2CYP3A4CYP2C19MAPT
SCHEMBL19783157 0.79 KMT2A (0.60) KMT2ACYP1A2CYP3A4CYP2C19PDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 381 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109485620-A A kind of preparation method of 2- methoxyl group -6- methoxybenzothiazole 安徽工大化工科技有限公司 2019-03-19 CN claimed
CN-109456281-A A kind of preparation method of the chloro- 6- methoxybenzothiazole of 2- 安徽工大化工科技有限公司 2019-03-12 CN claimed
US-4826989-A Process for the preparation of luciferin compounds BOEHRINGER MANNHEIM GMBH (DE) 1989-05-02 US claimed
EP-0024525-B1 Process for the preparation of luciferin and its derivatives Roche Diagnostics GmbH (DE) 1982-06-30 EP claimed
EP-0024525-A1 Process for the preparation of luciferin and its derivatives Roche Diagnostics GmbH (DE) 1981-03-11 EP claimed
US-20260085073-A1 PYRAZOLYLCARBOXAMIDE COMPOUNDS AND THEIR USE IN THERAPY HOTSPOT THERAPEUTICS INC (US) 2026-03-26 US disclosed
CN-117120423-B Indolylamine 2, 3-dioxygenase inhibitors, methods of preparing the same, and pharmaceutical compositions containing the same 柳韩洋行 2026-02-27 CN disclosed
US-12528827-B2 Tricyclic heteroaryl-substituted quinoline and azaquinoline compounds as PAR4 inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2026-01-20 US disclosed
US-12378254-B2 Disubstituted octahydropyrrolo[3,4-c]pyrroles as orexin receptor modulators JANSSEN PHARMACEUTICA NV (BE) 2025-08-05 US disclosed
US-20250011293-A1 LEUKOTRIENE SYNTHESIS INHIBITORS NAEGIS PHARMACEUTICALS INC. (CA) 2025-01-09 US disclosed
US-12162871-B2 Inhibitors of VAP-1 ACUCELA INC. (US) 2024-12-10 US disclosed
US-20240309019-A1 TRICYCLIC HETEROARYL-SUBSTITUTED QUINOLINE AND AZAQUINOLINE COMPOUNDS AS PAR4 INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2024-09-19 US disclosed
EP-0742010-A2 Benzoquinolin-3-ones to inhibit bone loss ELI LILLY AND COMPANY (US) 1996-11-13 EP disclosed
EP-0733365-A2 Use of benzoquinolin-3-ones for the treatment and prevention of prostatic cancer ELI LILLY AND COMPANY (US) 1996-09-25 EP disclosed
US-5550134-A ADMINISTERING TO A MAMMAL FROM A SERIES OF BENZOQUINOLIN-3-ONE COMPOUNDS ELI LILLY AND COMPANY (US) 1996-08-27 US disclosed
US-4873346-A BRONCHODILATORS, TREATMENT OF ASTHMA THE UPJOHN COMPANY (US) 1989-10-10 US disclosed
US-4826989-A Process for the preparation of luciferin compounds BOEHRINGER MANNHEIM GMBH (DE) 1989-05-02 US disclosed
EP-0123087-A1 Process for the preparation of heterocyclic phenyl ether CASSELLA Aktiengesellschaft (DE) 1984-10-31 EP disclosed
EP-0024525-B1 Process for the preparation of luciferin and its derivatives Roche Diagnostics GmbH (DE) 1982-06-30 EP disclosed
EP-0024525-A1 Process for the preparation of luciferin and its derivatives Roche Diagnostics GmbH (DE) 1981-03-11 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12162871-B2 Inhibitors of VAP-1 VAPB, VAPA, TOE1 KMT2A 4170/4885CYP1A2 4278/4885CYP3A4 4363/4885
US-20240309019-A1 TRICYCLIC HETEROARYL-SUBSTITUTED QUINOLINE AND AZAQUINOLINE COMPOUNDS AS PAR4 INHIBITORS F2RL3, PARP14, F2R KMT2A 897/4885CYP1A2 134/4885CYP3A4 24/4885
US-12378254-B2 Disubstituted octahydropyrrolo[3,4-c]pyrroles as orexin receptor modulators HCRTR2, HCRTR1, OXTR KMT2A 1722/4885CYP1A2 2758/4885CYP3A4 2368/4885
US-20260085073-A1 PYRAZOLYLCARBOXAMIDE COMPOUNDS AND THEIR USE IN THERAPY MALT1, BCL6, BCL3 KMT2A 2239/4885CYP1A2 3089/4885CYP3A4 2504/4885
US-12528827-B2 Tricyclic heteroaryl-substituted quinoline and azaquinoline compounds as PAR4 inhibitors F2RL3, F2R, PF4 KMT2A 2733/4885CYP1A2 103/4885CYP3A4 23/4885
US-20250011293-A1 LEUKOTRIENE SYNTHESIS INHIBITORS LTC4S, LTB4R2, LTA4H KMT2A 4046/4885CYP1A2 502/4885CYP3A4 624/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.