SCHEMBL14499486

SCHEMBL14499486

CC(=O)OCOC(=O)Cc1ccc(C)cc1F

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.39
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 1/20 0.38
HSD17B10 Q99714 1/20 0.38
SMN1; SMN2 Q16637 3/20 0.36
LMNA P02545 3/20 0.36
SRC P12931 1/20 0.36
MTNR1A P48039 1/20 0.35
MTNR1B P49286 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
KDM5A P29375 1/20 0.35
KDM4C Q9H3R0 1/20 0.35
KDM5B Q9UGL1 1/20 0.35
MYC P01106 1/20 0.35
MEN1 O00255 2/20 0.34
POLB P06746 2/20 0.34
KMT2A Q03164 2/20 0.34
GAA P10253 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
MAOB P27338 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10258195 0.86 NLRP3 (0.43) P2RX7ALDH1A1HSD17B10SMN1; SMN2L3MBTL1
SCHEMBL14194529 0.85 CHRNA7 (0.41) ALDH1A1KDM4ESMN1; SMN2MTNR1AMTNR1B
SCHEMBL4513880 0.84 ALDH1A1 (0.37) ALDH1A1KDM4ESMN1; SMN2LMNAMTNR1A
SCHEMBL2403273 0.82 L3MBTL1 (0.40) P2RX7ALDH1A1KDM4EHSD17B10SMN1; SMN2
SCHEMBL13949103 0.81 P2RX7 (0.45) P2RX7ALDH1A1KDM4EHSD17B10LMNA
SCHEMBL10862456 0.79 P2RX7 (0.45) P2RX7SMN1; SMN2LMNASRCKDM5A
SCHEMBL14499487 0.78 P2RX7 (0.44) P2RX7HSD17B10KDM5AKDM4CKDM5B
SCHEMBL14223664 0.78 MCL1 (0.40) ALDH1A1
SCHEMBL5545008 0.75 SRC (0.59) P2RX7ALDH1A1KDM4ESMN1; SMN2SRC
SCHEMBL15777939 0.74 P2RX7 (0.42) P2RX7ALDH1A1HSD17B10SMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7226951-B2 Compounds having selective cytochrome P450RAI-1 or selective cytochrome P450RAI-2 inhibitory activity and methods of obtaining the same ALLERGAN, INC. (US) 2007-06-05 US disclosed