SCHEMBL14565737

SCHEMBL14565737

O=CNC1CCCN(S(=O)(=O)c2ccc(Cl)c(Cl)c2)CC1=O

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.47
KDM4E B2RXH2 1/20 0.47
POLB P06746 1/20 0.47
VCAM1 P19320 1/20 0.43
NPBWR1 P48145 1/20 0.43
MCHR1 Q99705 1/20 0.43
TSHR P16473 4/20 0.42
CTSG P08311 2/20 0.41
CMA1 P23946 2/20 0.41
RECQL P46063 1/20 0.41
HCRTR1 O43613 1/20 0.41
HCRTR2 O43614 1/20 0.41
MAPK1 P28482 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
MCOLN3 Q8TDD5 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
HTR7 P34969 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14565729 0.82 PKM (0.46) KDM4EMEN1KMT2A
SCHEMBL14565739 0.81 GPBAR1 (0.56) POLBTSHRMAPK1MEN1KMT2A
SCHEMBL5444937 0.80 KDM4E (0.52) RAB9AKDM4EPOLBVCAM1NPBWR1
SCHEMBL14565751 0.75 TSHR (0.36) POLBTSHRMAPK1MEN1KMT2A
SCHEMBL14565738 0.74 KMT2A (0.48) TSHRMEN1KMT2AL3MBTL1
SCHEMBL494192 0.74 KDM4E (0.74) RAB9AKDM4EPOLBVCAM1NPBWR1
SCHEMBL14565744 0.74 PKM (0.49) RAB9AKDM4EPOLBTSHRMAPK1
SCHEMBL14565752 0.73 POLB (0.37) KDM4EPOLBTSHRMAPK1MEN1
SCHEMBL14565734 0.73 CTSK (0.49)
SCHEMBL14565743 0.73 MEN1 (0.55) TSHRHCRTR1HCRTR2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7196099-B2 Compounds and compositions as cathepsin inhibitors AVENTIS PHARMACEUTICALS INC. (US) 2007-03-27 US disclosed