Zenidolol

Zenidolol

SCHEMBL146178

Cc1ccc(OCC(O)C(C)NC(C)C)c2c1CCC2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 7/20 1.00
ADRB1 P08588 5/20 1.00
ADRB3 P13945 3/20 1.00
CYP2D6 P10635 2/20 1.00
TSHR P16473 2/20 1.00
KDM4E B2RXH2 2/20 1.00
ADRA2A P08913 1/20 1.00
TP53 P04637 1/20 1.00
CYP1A2 P05177 1/20 1.00
CYP3A4 P08684 1/20 1.00
NFKB1 P19838 1/20 1.00
HIF1A Q16665 1/20 1.00
NPSR1 Q6W5P4 2/20 0.97
MEN1 O00255 1/20 0.97
LMNA P02545 1/20 0.97
PMP22 Q01453 1/20 0.97
KMT2A Q03164 1/20 0.97
RXRG P48443 7/20 0.44
RXRA P19793 6/20 0.44
RXRB P28702 6/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Zenidolol SCHEMBL29558331 1.00 ADRB2 (1.00) ADRB2ADRB1ADRB3CYP2D6TSHR
Zenidolol SCHEMBL8027938 1.00 ADRB2 (1.00) ADRB2ADRB1ADRB3CYP2D6TSHR
Zenidolol SCHEMBL14941581 1.00 ADRB2 (1.00) ADRB2ADRB1ADRB3CYP2D6TSHR
Zenidolol SCHEMBL15058356 1.00 ADRB2 (1.00) ADRB2ADRB1ADRB3CYP2D6TSHR
Zenidolol SCHEMBL29387637 1.00 ADRB2 (1.00) ADRB2ADRB1ADRB3CYP2D6TSHR
Zenidolol SCHEMBL5485188 0.99 ADRB2 (1.00) ADRB2ADRB1ADRB3CYP2D6TSHR
Zenidolol SCHEMBL29686378 0.99 ADRB2 (1.00) ADRB2ADRB1ADRB3CYP2D6TSHR
Zenidolol SCHEMBL31074300 0.99 ADRB2 (1.00) ADRB2ADRB1ADRB3CYP2D6TSHR
SCHEMBL15549338 0.85 ADRB2 (0.74) ADRB2ADRB1ADRB3CYP2D6TSHR
SCHEMBL11266032 0.85 ADRB2 (0.74) ADRB2ADRB1ADRB3CYP2D6TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 650 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10788500-B2 IL1RL-1 as a cardiovascular disease marker and therapeutic target BRIGHAM & WOMEN'S HOSPITAL, INC. (US) 2020-09-29 US claimed
US-20180217160-A1 IL1RL-1 as a Cardiovascular Disease Marker and Therapeutic Target THE BRIGHAM & WOMEN'S HOSPITAL, INC. 2018-08-02 US claimed
EP-3072978-B1 1L1RL-1 AS A CARDIOVASCULAR DISEASE MARKER BRIGHAM & WOMENS HOSPITAL INC (US) 2018-07-11 EP claimed
US-9851362-B2 1L1RL-1 as a cardiovascular disease marker and therapeutic target The Brigham & Women's Hosptial, Inc. (US) 2017-12-26 US claimed
EP-3072978-A1 1L1RL-1 AS A CARDIOVASCULAR DISEASE MARKER AND THERAPEUTIC TARGET The Brigham and Women's Hospital, Inc. (US) 2016-09-28 EP claimed
EP-2336359-B1 1L1RL-1 as a cardiovascular disease marker BRIGHAM & WOMENS HOSPITAL (US) 2016-04-20 EP claimed
US-20150153360-A1 1L1RL-1 as a Cardiovascular Disease Marker and Therapeutic Target THE BRIGHAM AND WOMEN'S HOSPITAL, INC. (US) 2015-06-04 US claimed
US-20140357724-A1 BETA 2 ADRENOCEPTOR ANTAGONISTS FOR TREATING ORTHOSTATIC HYPOTENSION INDIANA UNIVERSITY RESEARCH & TECHNOLOGY CORPORATION (US) 2014-12-04 US claimed
WO-2014063189-A1 METHODS AND PRODUCTS FOR PREVENTING AND/OR TREATING A STRESS INDUCED CARDIOMYOPATHY ADELAIDE RESEARCH & INNOVATION PTY LTD (AU) 2014-05-01 WO claimed
US-20120244208-A1 COSMETIC SKIN CARE METHODS AND COMPOSITIONS de Villiers, Malan (ZA) 2012-09-27 US claimed
EP-0209897-A2 Peptide enzyme inhibitors MERCK & CO. INC. (US) 1987-01-28 EP claimed
EP-0163237-A2 Di- and tri-peptidal renin inhibitors MERCK & CO. INC. (US) 1985-12-04 EP claimed
EP-0157409-A2 Renin inhibitors containing 2-substituted statine MERCK & CO. INC. (US) 1985-10-09 EP claimed
EP-0156318-A2 C-terminal amide cyclic renin inhibitors containing peptide isosteres MERCK & CO. INC. (US) 1985-10-02 EP claimed
EP-0156322-A2 Renin inhibitors containing peptide isosteres MERCK & CO. INC. (US) 1985-10-02 EP claimed
EP-0129189-A2 Renin inhibitors containing a C-terminal amide cycle and compositions and combinations containing the same MERCK & CO. INC. (US) 1984-12-27 EP claimed
EP-0105996-A1 Ophthalmic compositions for treating elevated intraocular pressure MERCK & CO. INC. (US) 1984-04-25 EP claimed
EP-0003664-B1 ALKANOLAMINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1982-02-17 EP claimed
US-4275058-A 1-(7-METHYLINDAN-4-YLOXY)-3-ISOPROPYLAMINOBUTAN-2-OL IMPERIAL CHEMICAL INDUSTRIES LIMITED (GB) 1981-06-23 US claimed
EP-0003664-A1 Alkanolamine derivatives, process for their preparation and pharmaceutical compositions containing them IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1979-08-22 EP claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140357724-A1 BETA 2 ADRENOCEPTOR ANTAGONISTS FOR TREATING ORTHOSTATIC HYPOTENSION ADRB2, ADRA2C, ADRA2A ADRB2 1/4885ADRB1 6/4885ADRB3 5/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.