Zenidolol

Zenidolol

SCHEMBL29686378

Cc1ccc(OC[C@H](O)[C@@H](C)NC(C)C)c2c1CCC2.Cl

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABL1ACEACHEACVR1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALKAVPR1AAVPR2BCHEBCRCA2CACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCASRCCR5CDK4CDK6CFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNA3CHRNA7CHRNB1CHRNB4CHRNDCHRNECHRNGCOXFA4COXFA4L2CRBNCSF1RCUL4ACYP19A1DDB1DPP4DRD1DRD2DRD3DRD4EDNRAEGFREML4ERBB2ERBB4ESR1ESR2FGFR1FGFR3FLT1FLT3FLT4GAAGABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGHSRGLAGNRHRGPD2GRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BGSTP1HCN4HCRTR1HCRTR2HDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HRH2HRH3HSD11B1HSP90AA1HSP90AB1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IMPDH1IMPDH2ITGA2BITGB3ITKJAK1JAK2KCNA1KCNA10KCNA2KCNA3KCNA4KCNA5KCNA6KCNA7KCNB1KCNB2KCNC1KCNC2KCNC3KCNC4KCND1KCND2KCND3KCNF1KCNG1KCNG2KCNG3KCNG4KCNH1KCNH2KCNH3KCNH4KCNH5KCNH6KCNH7KCNH8KCNJ2KCNJ3KCNJ5KCNK3KCNK9KCNQ1KCNQ2KCNQ3KCNQ4KCNQ5KCNS1KCNS2KCNS3KCNV1KCNV2KDRKITKLKB1LCKMMAOAMAOBMAPK14METMMP1MMP13MMP7MMP8MT-ND1MT-ND2MT-ND3MT-ND4MT-ND4LMT-ND5MT-ND6NDUFA1NDUFA10NDUFA11NDUFA12NDUFA13NDUFA2NDUFA3NDUFA5NDUFA6NDUFA7NDUFA8NDUFA9NDUFAB1NDUFAF1NDUFAF2NDUFAF3NDUFAF4NDUFB1NDUFB10NDUFB11NDUFB2NDUFB3NDUFB4NDUFB5NDUFB6NDUFB7NDUFB8NDUFB9NDUFC1NDUFC2NDUFS1NDUFS2NDUFS3NDUFS4NDUFS5NDUFS6NDUFS7NDUFS8NDUFV1NDUFV2NDUFV3NR3C1NS5ANTRK1NTRK2NTRK3ODC1OPRD1OPRK1OPRM1P2RY12PAHPARP1PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDE5APDE7APDE7BPDE8APDE8BPDGFRAPDGFRBPIK3CAPIK3CDPNPPOLA1POLA2POLD1POLD2POLD3POLD4POLEPOLE2POLE3PPARGPRIM1PRIM2PRKCAPRKCBPRKCDPRKCEPRKCGPRKCHPRKCIPRKCQPRKCZPRKD1PRKD3PTGS1PTGS2RBX1RENRETROCK1ROCK2RPE65RRM1RRM2RRM2BS1PR1S1PR2S1PR3S1PR4S1PR5SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC18A2SLC6A1SLC6A2SLC6A3SLC6A4SLC9A3SRCTACR1TOP1TOP2ATOP2BTTRTYMPdacAdacBdacCembAfolAftsIgyrAgyrBmrcAmrcBmrdAparCparEpolrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Zenidolol. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 known ✓ P07550 6/20 1.00
ADRB1 known ✓ P08588 5/20 0.97
ADRB3 known ✓ P13945 3/20 0.97
ADRA2A known ✓ P08913 1/20 0.97
HTR1A known ✓ P08908 1/20 0.35
SLC6A4 known ✓ P31645 1/20 0.35
SIGMAR1 known ✓ Q99720 1/20 0.35
NPSR1 Q6W5P4 2/20 1.00
MEN1 O00255 1/20 1.00
LMNA P02545 1/20 1.00
PMP22 Q01453 1/20 1.00
KMT2A Q03164 1/20 1.00
CYP2D6 P10635 2/20 0.97
TSHR P16473 2/20 0.97
KDM4E B2RXH2 2/20 0.97
TP53 P04637 1/20 0.97
CYP1A2 P05177 1/20 0.97
CYP3A4 P08684 1/20 0.97
NFKB1 P19838 1/20 0.97
HIF1A Q16665 1/20 0.97

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Zenidolol SCHEMBL31074300 1.00 ADRB2 (1.00) ADRB2NPSR1MEN1LMNAPMP22
Zenidolol SCHEMBL5485188 1.00 ADRB2 (1.00) ADRB2NPSR1MEN1LMNAPMP22
Zenidolol SCHEMBL146178 0.99 ADRB2 (1.00) ADRB2NPSR1MEN1LMNAPMP22
Zenidolol SCHEMBL29387637 0.99 ADRB2 (1.00) ADRB2NPSR1MEN1LMNAPMP22
Zenidolol SCHEMBL29558331 0.99 ADRB2 (1.00) ADRB2NPSR1MEN1LMNAPMP22
Zenidolol SCHEMBL14941581 0.99 ADRB2 (1.00) ADRB2NPSR1MEN1LMNAPMP22
Zenidolol SCHEMBL8027938 0.99 ADRB2 (1.00) ADRB2NPSR1MEN1LMNAPMP22
Zenidolol SCHEMBL15058356 0.99 ADRB2 (1.00) ADRB2NPSR1MEN1LMNAPMP22
SCHEMBL15549338 0.84 ADRB2 (0.74) ADRB2NPSR1MEN1LMNAPMP22
SCHEMBL11266032 0.84 ADRB2 (0.74) ADRB2NPSR1MEN1LMNAPMP22

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4048809-B1 SYSTEMS AND METHODS FOR PREDICTING THERAPEUTIC SENSITIVITY TEMPUS AI INC (US) 2026-05-27 EP disclosed
EP-4729940-A2 LARGE SCALE ORGANOID ANALYSIS Tempus AI, Inc. (US) 2026-04-22 EP disclosed
US-20260011445-A1 SYSTEMS AND METHODS FOR PREDICTING THERAPEUTIC SENSITIVITY TEMPUS AI INC (US) 2026-01-08 US disclosed
EP-4070098-B1 LARGE SCALE ORGANOID ANALYSIS TEMPUS AI INC (US) 2025-12-24 EP disclosed
US-12451250-B2 Systems and methods for predicting therapeutic sensitivity TEMPUS AI, INC. (US) 2025-10-21 US disclosed
US-11759445-B2 Use of Rivastigmine in preparation of anti-radiation medicament SOOCHOW UNIVERSITY (CN) 2023-09-19 US disclosed
US-20220392640-A1 SYSTEMS AND METHODS FOR PREDICTING THERAPEUTIC SENSITIVITY TEMPUS AI, INC. 2022-12-08 US disclosed
US-20220341914-A1 LARGE SCALE ORGANOID ANALYSIS TEMPUS AI, INC. (F/K/A TEMPUS LABS, INC.) 2022-10-27 US disclosed
US-11415571-B2 Large scale organoid analysis TEMPUS LABS, INC. (US) 2022-08-16 US disclosed
US-20220175714-A1 USE OF RIVASTIGMINE IN PREPARATION OF ANTI-RADIATION MEDICAMENT SOOCHOW UNIVERSITY (CN) 2022-06-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260011445-A1 SYSTEMS AND METHODS FOR PREDICTING THERAPEUTIC SENSITIVITY BRCA1, PARP2, PARP4 ADRB2 3687/4885ADRB1 3784/4885ADRB3 3735/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.