SCHEMBL1462095

SCHEMBL1462095

Nc1c(F)ccc(CCCS(N)(=O)=O)c1Cl

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CA2 P00918 3/20 0.37
RECQL P46063 1/20 0.34
CA1 P00915 1/20 0.33
CA9 Q16790 1/20 0.33
PTGES2 Q9H7Z7 2/20 0.31
PTGS1 P23219 1/20 0.31
PTGS2 P35354 1/20 0.31
SOS1 Q07889 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8215818 0.84 CA2 (0.39) CA2RECQLCA1
SCHEMBL1462274 0.74 TAAR1 (0.37) CA2RECQLCA1CA9PTGES2
SCHEMBL1492045 0.68 RECQL (0.40) CA2RECQLCA1CA9PTGES2
SCHEMBL1494448 0.65 MGLL (0.37) CA2RECQLCA1CA9PTGES2
SCHEMBL2777071 0.64 TNF (0.38) CA2CA1CA9
SCHEMBL1462138 0.63 BRAF (0.46) PTGES2
SCHEMBL25437680 0.62 MGLL (0.62) CA2CA1CA9
SCHEMBL15924708 0.62 TAAR1 (0.53) CA2CA1CA9
SCHEMBL14784534 0.62 MAPK1 (0.43) CA2CA1CA9
SCHEMBL3238785 0.61 PSEN1 (0.42) CA2CA1CA9PTGES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2493865-A2 RAF INHIBITOR COMPOUNDS AND METHODS OF USE THEREOF Array Biopharma, Inc. (US) 2012-09-05 EP disclosed
WO-2011025938-A2 RAF INHIBITOR COMPOUNDS AND METHODS OF USE THEREOF ARRAY BIOPHARMA INC. (US) 2011-03-03 WO disclosed