SCHEMBL8215818

SCHEMBL8215818

Nc1c(F)ccc(CCCS(N)(=O)=O)c1F

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CA2 P00918 4/20 0.39
RECQL P46063 1/20 0.36
NOS1 P29475 1/20 0.32
MGLL Q99685 1/20 0.31
CA12 O43570 1/20 0.30
CA1 P00915 1/20 0.30
CA7 P43166 1/20 0.30
CA13 Q8N1Q1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1462095 0.84 CA2 (0.37) CA2RECQLCA1
SCHEMBL1494448 0.73 MGLL (0.37) CA2RECQLMGLLCA12CA1
SCHEMBL1492045 0.73 RECQL (0.40) CA2RECQLCA12CA1CA7
SCHEMBL1462230 0.71 CA2 (0.30) CA2
SCHEMBL671337 0.68 LOXL2 (0.39)
SCHEMBL29467988 0.68 LOXL2 (0.39)
SCHEMBL25437680 0.65 MGLL (0.62) CA2MGLLCA12CA1
SCHEMBL15924708 0.65 TAAR1 (0.53) CA2MGLLCA12CA1
SCHEMBL28452491 0.64 APLNR (0.49) CA2CA12CA1CA7
SCHEMBL16058359 0.63 CA2 (0.45) CA2CA12CA1CA7CA13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2470511-A1 RAF INHIBITOR COMPOUNDS AND METHODS OF USE THEREOF Genentech, Inc. (US) 2012-07-04 EP disclosed
WO-2011025965-A1 RAF INHIBITOR COMPOUNDS AND METHODS OF USE THEREOF GENENTECH, INC. (US) 2011-03-03 WO disclosed