SCHEMBL14664339

SCHEMBL14664339

COc1cccc2nc(-c3ccc([N+](=O)[O-])o3)[nH]c12

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 1/20 0.60
MMP9 P14780 1/20 0.60
MMP8 P22894 1/20 0.60
MMP13 P45452 1/20 0.60
AMY1A P0DUB6 3/20 0.40
ILK Q13418 1/20 0.39
TNKS O95271 1/20 0.38
TNKS2 Q9H2K2 1/20 0.38
PARP2 Q9UGN5 1/20 0.38
SLC2A1 P11166 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
TP53 P04637 1/20 0.37
CYP1A2 P05177 1/20 0.37
BRCA1 P38398 1/20 0.37
HNF4A P41235 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
HIF1A Q16665 1/20 0.37
MITF O75030 1/20 0.37
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14664340 0.87 MMP2 (0.57) MMP2MMP9MMP8MMP13SLC2A1
SCHEMBL12713529 0.84 MMP2 (0.64) MMP2MMP9MMP8MMP13SLC2A1
SCHEMBL1609480 0.81 MMP2 (0.64) MMP2MMP9MMP8MMP13TNKS
SCHEMBL10694677 0.76 MMP2 (1.00) MMP2MMP9MMP8MMP13NPC1
SCHEMBL9044504 0.76 GUSB (0.56) AMY1AALDH1A1TDP1GUSB
SCHEMBL28027631 0.69 TNKS (0.54) AMY1ATNKSTNKS2PARP2NPC1
SCHEMBL10691037 0.69 MMP2 (0.68) MMP2MMP9MMP8MMP13SLC2A1
SCHEMBL10688373 0.69 MMP2 (0.68) MMP2MMP9MMP8MMP13AMY1A
SCHEMBL30360160 0.69 MMP2 (0.68) MMP2MMP9MMP8MMP13AMY1A
SCHEMBL4420447 0.68 NQO2 (0.46) AMY1ANPC1RAB9ATP53SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9617249-B2 Benzoheterocyclic anti-bacterial agents UNIVERSITY OF NOTRE DAME DU LAC (US) 2017-04-11 US disclosed
US-9617249-B2 Benzoheterocyclic anti-bacterial agents UNIVERSITY OF NOTRE DAME DU LAC (US) 2017-04-11 US disclosed
US-8362268-B2 Anti-bacterial agents from benzo[d]heterocyclic scaffolds for prevention and treatment of multidrug resistant bacteria UNIVERSITY OF NOTRE DAME DU LAC (US) 2013-01-29 US disclosed
US-8362268-B2 Anti-bacterial agents from benzo[d]heterocyclic scaffolds for prevention and treatment of multidrug resistant bacteria UNIVERSITY OF NOTRE DAME DU LAC (US) 2013-01-29 US disclosed