SCHEMBL14722369

SCHEMBL14722369

CC(C)(C)OC(=O)NC1CN(c2ncc(C(=O)N(C3CC3)C3CCN(Cc4ccccc4)CC3)cn2)CC1c1cc(F)c(F)cc1F

nearest known ligand 0.42

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 14/20 0.42
CHRM2 P08172 6/20 0.40
CHRM1 P11229 5/20 0.40
CHRM3 P20309 4/20 0.39
CHRM5 P08912 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14723328 0.86 GPR119 (0.39)
SCHEMBL6128140 0.85 GPR119 (0.36)
SCHEMBL14722228 0.85 PDE4B (0.42)
SCHEMBL14730335 0.80 DPP4 (0.38)
SCHEMBL14730281 0.79 MAOA (0.32)
SCHEMBL14730229 0.79 GPR119 (0.40)
SCHEMBL14722672 0.79 GPR119 (0.40)
SCHEMBL6128597 0.79 GPR119 (0.40)
SCHEMBL14722527 0.79 PDE4B (0.41)
SCHEMBL147896 0.78 L3MBTL1 (0.46) CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013026587-A1 1,4 DISUBSTITUTED PYRROLIDINE - 3 - YL -AMINE DERIVATIVES AND THEIR USE FOR THE TREATMENT OF METABOLIC DISORDERS PROSIDION LIMITED (GB) 2013-02-28 WO disclosed