SCHEMBL14765127

SCHEMBL14765127

CCCc1nnc2c(C)nc3ccccc3n12

nearest known ligand 0.59

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 7/20 0.53
PDE10A Q9Y233 5/20 0.53
HTR2C P28335 1/20 0.53
POLB P06746 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14354843 0.90 POLB (0.54) PDE2APDE10AHTR2CPOLBNPSR1
SCHEMBL7342631 0.84 TYMS (0.56) HTR2CPOLBNPSR1
SCHEMBL10844192 0.81 ALOX15 (0.60) HTR2CPOLBNPSR1
SCHEMBL971822 0.79 PDE10A (0.63) PDE2APDE10A
SCHEMBL14765137 0.77 PDE2A (0.56) PDE2APDE10AHTR2C
SCHEMBL7347836 0.76 NPSR1 (0.54) HTR2CPOLBNPSR1
SCHEMBL14764825 0.76 PDE10A (0.58) PDE2APDE10A
SCHEMBL14054782 0.75 PDE2A (0.67) PDE2APDE10APOLB
SCHEMBL7345568 0.75 ALDH1A1 (0.69) HTR2C
SCHEMBL28574640 0.75 KDM4E (0.78) POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013034755-A1 TRIAZOLOPYRAZINE DERIVATIVES AND THEIR USE FOR TREATING NEUROLOGICAL AND PSYCHIATRIC DISORDERS H. LUNDBECK A/S (DK) 2013-03-14 WO claimed
WO-2013034755-A1 TRIAZOLOPYRAZINE DERIVATIVES AND THEIR USE FOR TREATING NEUROLOGICAL AND PSYCHIATRIC DISORDERS H. LUNDBECK A/S (DK) 2013-03-14 WO disclosed
WO-2013034755-A1 TRIAZOLOPYRAZINE DERIVATIVES AND THEIR USE FOR TREATING NEUROLOGICAL AND PSYCHIATRIC DISORDERS H. LUNDBECK A/S (DK) 2013-03-14 WO disclosed