SCHEMBL14769272

SCHEMBL14769272

CCOC(=O)c1ccc(OC[C@@H]2C[C@@H](OB(N)O)CN2C)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41
STS P08842 1/20 0.39
TBXAS1 P24557 1/20 0.39
CHRNB2 P17787 1/20 0.39
CHRNA5 P30532 1/20 0.39
CHRNA7 P36544 1/20 0.39
CHRNA4 P43681 1/20 0.39
KMT2A Q03164 1/20 0.39
LMNA P02545 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
MAOA P21397 1/20 0.39
TDP1 Q9NUW8 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
MAPT P10636 1/20 0.37
MMP13 P45452 1/20 0.37
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL85313 0.81 KCNH2 (0.46) KCNH2HRH3STSTBXAS1CHRNB2
SCHEMBL14592630 0.74 EPHX2 (0.46) KCNH2HRH3STSKMT2ALMNA
SCHEMBL14592611 0.71 KCNJ1 (0.52) KCNH2CHRNB2CHRNA4KMT2ACYP1A2
SCHEMBL14592072 0.71 MAPT (0.52) CHRNB2CHRNA5CHRNA7CHRNA4KMT2A
SCHEMBL9384519 0.70 HRH3 (0.47) KCNH2HRH3TBXAS1CHRNB2CHRNA5
SCHEMBL13437495 0.69 TDP1 (0.41) KCNH2HRH3KMT2ATDP1L3MBTL1
SCHEMBL8536518 0.69 ALDH1A1 (0.51) KCNH2HRH3STSKMT2ALMNA
SCHEMBL9387166 0.68 LMNA (0.55) KCNH2HRH3CHRNB2CHRNA5CHRNA7
SCHEMBL27574704 0.68 CYP2C9 (0.54) KCNH2HRH3TBXAS1KMT2AMAOA
SCHEMBL85754 0.68 KCNH2 (0.44) KCNH2HRH3STSTBXAS1CHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130065882-A1 VLA-4 inhibitory drug MACHINAGA NOBUO (JP) 2013-03-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130065882-A1 VLA-4 inhibitory drug VCAM1, ITGB4, ITGA4 KCNH2 503/4885HRH3 372/4885STS 2041/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.