SCHEMBL14865107

SCHEMBL14865107

C=CC[C@@](O)(CCN[C@@H](C)c1ccc(-c2cccn(C)c2=O)cc1)c1ccc(F)cc1

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CASR P41180 1/20 0.34
ITGB1 P05556 1/20 0.33
ITGA4 P13612 1/20 0.33
ITGB7 P26010 1/20 0.33
OPRK1 P41145 2/20 0.32
APLNR P35414 1/20 0.32
HSD11B1 P28845 1/20 0.32
KMT2A Q03164 2/20 0.31
ROCK2 O75116 1/20 0.31
MITF O75030 1/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.31
HTT P42858 1/20 0.31
GPR139 Q6DWJ6 1/20 0.30
MC4R P32245 2/20 0.30
NPC1 O15118 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15959063 0.86 CASR (0.37) CASRITGB1ITGA4ITGB7OPRK1
SCHEMBL13638260 0.79 ALDH1A1 (0.35) CASRKMT2AMITFALDH1A1LMNA
SCHEMBL13953687 0.76 CASR (0.38) CASRKMT2AMITFALDH1A1LMNA
SCHEMBL957448 0.76 CASR (0.38) CASRKMT2AMITFALDH1A1LMNA
SCHEMBL15368397 0.73 GPR139 (0.35) ALDH1A1LMNAHTTGPR139
SCHEMBL13953572 0.73 MTNR1A (0.33) CASRKMT2AMITFALDH1A1LMNA
SCHEMBL13624881 0.72 LPL (0.40) KMT2AMITFALDH1A1LMNAMAPT
SCHEMBL13552181 0.71 HSD11B1 (0.47) HSD11B1
SCHEMBL1904136 0.70 HTT (0.35) CASRHSD11B1KMT2AMITFALDH1A1
SCHEMBL15959034 0.69 CASR (0.41) CASRHSD11B1KMT2AMITFALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2300461-B1 CYCLIC INHIBITORS OF 11BETA-HYDROXYSTEROID DEHYDROGENASE 1 VITAE PHARMACEUTICALS INC (US) 2013-04-17 EP disclosed