SCHEMBL1489101

SCHEMBL1489101

C=CCN(CC=C)OC(=O)ON(CC=C)CC=C

nearest known ligand 0.44

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.33
LMNA P02545 1/20 0.32
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
KDM4E B2RXH2 1/20 0.31
POLB P06746 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1489102 0.82 ALDH1A1 (0.38) ALDH1A1SMN1; SMN2LMNAMEN1KMT2A
SCHEMBL3469849 0.80 ALDH1A1 (0.37) ALDH1A1SMN1; SMN2MEN1KMT2AKDM4E
SCHEMBL612528 0.80 ALDH1A1 (0.37) ALDH1A1MEN1KMT2A
SCHEMBL169909 0.80 ALDH1A1 (0.37) ALDH1A1
SCHEMBL1257020 0.80 TSHR (0.40) ALDH1A1SMN1; SMN2LMNA
Hydrochloric Acid SCHEMBL28514951 0.78 ALDH1A1 (0.35) ALDH1A1MEN1KMT2A
SCHEMBL3453844 0.77 ALDH1A1 (0.34) ALDH1A1MEN1KMT2A
Acetic Acid SCHEMBL28451523 0.77 ALDH1A1 (0.34) ALDH1A1SMN1; SMN2LMNAMEN1KMT2A
SCHEMBL986380 0.77 ALDH1A1 (0.34) ALDH1A1
SCHEMBL2550182 0.77 ALDH1A1 (0.36) ALDH1A1LMNAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 25 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20150197484-A1 USE OF CANNABIDIOL PRODRUGS IN TOPICAL AND TRANSDERMAL ADMINISTRATION WITH MICRONEEDLES ZYNERBA PHARMACEUTICALS, INC. (US) 2015-07-16 US claimed
EP-2473475-A1 USE OF CANNABIDIOL PRODRUGS IN TOPICAL AND TRANSDERMAL ADMINISTRATION WITH MICRONEEDLES AllTranz Inc. (US) 2012-07-11 EP claimed
WO-2011026144-A1 USE OF CANNABIDIOL PRODRUGS IN TOPICAL AND TRANSDERMAL ADMINISTRATION WITH MICRONEEDLES ALLTRANZ INC. (US) 2011-03-03 WO claimed
US-20110052694-A1 USE OF CANNABIDIOL PRODRUGS IN TOPICAL AND TRANSDERMAL ADMINISTRATION WITH MICRONEEDLES ALLTRANZ INC. (US) 2011-03-03 US claimed
EP-2176208-A1 PRODRUGS OF CANNABIDIOL, COMPOSITIONS COMPRISING PRODRUGS OF CANNABIDIOL AND METHODS OF USING THE SAME AllTranz Inc. (US) 2010-04-21 EP claimed
US-20090036523-A1 PRODRUGS OF CANNABIDIOL, COMPOSITIONS COMPRISING PRODRUGS OF CANNABIDIOL AND METHODS OF USING THE SAME ALLTRANZ INC. (US) 2009-02-05 US claimed
WO-2009018389-A1 PRODRUGS OF CANNABIDIOL, COMPOSITIONS COMPRISING PRODRUGS OF CANNABIDIOL AND METHODS OF USING THE SAME ALLTRANZ INC. (US) 2009-02-05 WO claimed
US-11873272-B2 Antimicrobial and antiviral sulfur containing glycerol monoester derivatives Niche Biopharmaceuticals LLC (US) 2024-01-16 US disclosed
EP-4214191-A1 ANTIMICROBIAL AND ANTIVIRAL SULFUR CONTAINING GLYCEROL MONOESTER DERIVATIVES Niche Biopharmaceuticals LLC (US) 2023-07-26 EP disclosed
US-20230174473-A1 ANTIMICROBIAL AND ANTIVIRAL SULFUR CONTAINING GLYCEROL MONOESTER DERIVATIVES Niche Biopharmaceuticals LLC (US) 2023-06-08 US disclosed
US-11572342-B2 Antimicrobial and antiviral sulfur containing glycerol monoester derivatives Niche Biopharmaceuticals LLC (US) 2023-02-07 US disclosed
US-11365176-B2 Antimicrobial and antiviral sulfur containing glycerol monoester derivatives Niche Biopharmaceuticals LLC (US) 2022-06-21 US disclosed
US-20220127224-A1 ANTIMICROBIAL AND ANTIVIRAL SULFUR CONTAINING GLYCEROL MONOESTER DERIVATIVES Niche Biopharmaceuticals LLC 2022-04-28 US disclosed
US-8293786-B2 Prodrugs of cannabidiol, compositions comprising prodrugs of cannabidiol and methods of using the same ALLTRANZ INC. (US) 2012-10-23 US disclosed
EP-2473475-A1 USE OF CANNABIDIOL PRODRUGS IN TOPICAL AND TRANSDERMAL ADMINISTRATION WITH MICRONEEDLES AllTranz Inc. (US) 2012-07-11 EP disclosed
US-20110052694-A1 USE OF CANNABIDIOL PRODRUGS IN TOPICAL AND TRANSDERMAL ADMINISTRATION WITH MICRONEEDLES ALLTRANZ INC. (US) 2011-03-03 US disclosed
WO-2011026144-A1 USE OF CANNABIDIOL PRODRUGS IN TOPICAL AND TRANSDERMAL ADMINISTRATION WITH MICRONEEDLES ALLTRANZ INC. (US) 2011-03-03 WO disclosed
EP-2176208-A1 PRODRUGS OF CANNABIDIOL, COMPOSITIONS COMPRISING PRODRUGS OF CANNABIDIOL AND METHODS OF USING THE SAME AllTranz Inc. (US) 2010-04-21 EP disclosed
US-20090036523-A1 PRODRUGS OF CANNABIDIOL, COMPOSITIONS COMPRISING PRODRUGS OF CANNABIDIOL AND METHODS OF USING THE SAME ALLTRANZ INC. (US) 2009-02-05 US disclosed
WO-2009018389-A1 PRODRUGS OF CANNABIDIOL, COMPOSITIONS COMPRISING PRODRUGS OF CANNABIDIOL AND METHODS OF USING THE SAME ALLTRANZ INC. (US) 2009-02-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090036523-A1 PRODRUGS OF CANNABIDIOL, COMPOSITIONS COMPRISING PRODRUGS OF CANNABIDIOL AND METHODS OF USING THE SAME CNR2, CNR1, FAAH ALDH1A1 1490/4885SMN1; SMN2 2507/4885LMNA 1353/4885
US-20110052694-A1 USE OF CANNABIDIOL PRODRUGS IN TOPICAL AND TRANSDERMAL ADMINISTRATION WITH MICRONEEDLES PNLIP, CNR2, CNR1 ALDH1A1 3684/4885SMN1; SMN2 1670/4885LMNA 3547/4885
US-20220127224-A1 ANTIMICROBIAL AND ANTIVIRAL SULFUR CONTAINING GLYCEROL MONOESTER DERIVATIVES MAVS, SARS1, MGLL ALDH1A1 3686/4885SMN1; SMN2 3535/4885LMNA 4761/4885
US-11572342-B2 Antimicrobial and antiviral sulfur containing glycerol monoester derivatives MAVS, SARS1, MGLL ALDH1A1 3686/4885SMN1; SMN2 3535/4885LMNA 4761/4885
US-11873272-B2 Antimicrobial and antiviral sulfur containing glycerol monoester derivatives MAVS, SARS1, MGLL ALDH1A1 3686/4885SMN1; SMN2 3535/4885LMNA 4761/4885
US-20230174473-A1 ANTIMICROBIAL AND ANTIVIRAL SULFUR CONTAINING GLYCEROL MONOESTER DERIVATIVES MAVS, SARS1, MGLL ALDH1A1 3686/4885SMN1; SMN2 3535/4885LMNA 4761/4885
US-20150197484-A1 USE OF CANNABIDIOL PRODRUGS IN TOPICAL AND TRANSDERMAL ADMINISTRATION WITH MICRONEEDLES PNLIP, CNR2, CNR1 ALDH1A1 3684/4885SMN1; SMN2 1670/4885LMNA 3547/4885
US-11365176-B2 Antimicrobial and antiviral sulfur containing glycerol monoester derivatives MAVS, SARS1, MGLL ALDH1A1 3686/4885SMN1; SMN2 3535/4885LMNA 4761/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.