SCHEMBL1489102

SCHEMBL1489102

C=CCN(CC=C)OC(=O)O

nearest known ligand 0.41

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.36
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
KDM4E B2RXH2 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1489101 0.82 ALDH1A1 (0.44) ALDH1A1LMNAMEN1KMT2AKDM4E
Acetic Acid SCHEMBL28451523 0.79 ALDH1A1 (0.34) ALDH1A1LMNAMEN1KMT2AKDM4E
SCHEMBL169909 0.78 ALDH1A1 (0.37) ALDH1A1TSHR
SCHEMBL3469849 0.78 ALDH1A1 (0.37) ALDH1A1MEN1KMT2AKDM4ESMN1; SMN2
SCHEMBL1257020 0.78 TSHR (0.40) ALDH1A1LMNASMN1; SMN2TSHR
SCHEMBL612528 0.78 ALDH1A1 (0.37) ALDH1A1MEN1KMT2ATSHR
Hydrochloric Acid SCHEMBL28514951 0.76 ALDH1A1 (0.35) ALDH1A1MEN1KMT2ATSHR
SCHEMBL10784897 0.76 KDM4E (0.33) ALDH1A1MEN1KMT2AKDM4ESMN1; SMN2
SCHEMBL3453844 0.75 ALDH1A1 (0.34) ALDH1A1MEN1KMT2A
SCHEMBL986380 0.75 ALDH1A1 (0.34) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 28 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20150197484-A1 USE OF CANNABIDIOL PRODRUGS IN TOPICAL AND TRANSDERMAL ADMINISTRATION WITH MICRONEEDLES ZYNERBA PHARMACEUTICALS, INC. (US) 2015-07-16 US claimed
EP-2473475-A1 USE OF CANNABIDIOL PRODRUGS IN TOPICAL AND TRANSDERMAL ADMINISTRATION WITH MICRONEEDLES AllTranz Inc. (US) 2012-07-11 EP claimed
US-20110052694-A1 USE OF CANNABIDIOL PRODRUGS IN TOPICAL AND TRANSDERMAL ADMINISTRATION WITH MICRONEEDLES ALLTRANZ INC. (US) 2011-03-03 US claimed
WO-2011026144-A1 USE OF CANNABIDIOL PRODRUGS IN TOPICAL AND TRANSDERMAL ADMINISTRATION WITH MICRONEEDLES ALLTRANZ INC. (US) 2011-03-03 WO claimed
EP-2176208-A1 PRODRUGS OF CANNABIDIOL, COMPOSITIONS COMPRISING PRODRUGS OF CANNABIDIOL AND METHODS OF USING THE SAME AllTranz Inc. (US) 2010-04-21 EP claimed
US-20090036523-A1 PRODRUGS OF CANNABIDIOL, COMPOSITIONS COMPRISING PRODRUGS OF CANNABIDIOL AND METHODS OF USING THE SAME ALLTRANZ INC. (US) 2009-02-05 US claimed
WO-2009018389-A1 PRODRUGS OF CANNABIDIOL, COMPOSITIONS COMPRISING PRODRUGS OF CANNABIDIOL AND METHODS OF USING THE SAME ALLTRANZ INC. (US) 2009-02-05 WO claimed
US-11873272-B2 Antimicrobial and antiviral sulfur containing glycerol monoester derivatives Niche Biopharmaceuticals LLC (US) 2024-01-16 US disclosed
EP-4214191-A1 ANTIMICROBIAL AND ANTIVIRAL SULFUR CONTAINING GLYCEROL MONOESTER DERIVATIVES Niche Biopharmaceuticals LLC (US) 2023-07-26 EP disclosed
CN-116323556-A Antimicrobial and antiviral sulfur-containing monoglyceride derivatives 尼奇生物制药有限责任公司 2023-06-23 CN disclosed
US-20230174473-A1 ANTIMICROBIAL AND ANTIVIRAL SULFUR CONTAINING GLYCEROL MONOESTER DERIVATIVES Niche Biopharmaceuticals LLC (US) 2023-06-08 US disclosed
US-11572342-B2 Antimicrobial and antiviral sulfur containing glycerol monoester derivatives Niche Biopharmaceuticals LLC (US) 2023-02-07 US disclosed
US-11365176-B2 Antimicrobial and antiviral sulfur containing glycerol monoester derivatives Niche Biopharmaceuticals LLC (US) 2022-06-21 US disclosed
WO-2011026144-A1 USE OF CANNABIDIOL PRODRUGS IN TOPICAL AND TRANSDERMAL ADMINISTRATION WITH MICRONEEDLES ALLTRANZ INC. (US) 2011-03-03 WO disclosed
US-20110052694-A1 USE OF CANNABIDIOL PRODRUGS IN TOPICAL AND TRANSDERMAL ADMINISTRATION WITH MICRONEEDLES ALLTRANZ INC. (US) 2011-03-03 US disclosed
EP-2176208-A1 PRODRUGS OF CANNABIDIOL, COMPOSITIONS COMPRISING PRODRUGS OF CANNABIDIOL AND METHODS OF USING THE SAME AllTranz Inc. (US) 2010-04-21 EP disclosed
US-20090036523-A1 PRODRUGS OF CANNABIDIOL, COMPOSITIONS COMPRISING PRODRUGS OF CANNABIDIOL AND METHODS OF USING THE SAME ALLTRANZ INC. (US) 2009-02-05 US disclosed
WO-2009018389-A1 PRODRUGS OF CANNABIDIOL, COMPOSITIONS COMPRISING PRODRUGS OF CANNABIDIOL AND METHODS OF USING THE SAME ALLTRANZ INC. (US) 2009-02-05 WO disclosed
EP-0842142-A1 PROCESS FOR PRODUCING $g(a)-(N,N DIALKYL)-AMINO CARBOXYLIC ACID AMIDES BASF AKTIENGESELLSCHAFT (DE) 1998-05-20 EP disclosed
WO-1997005096-A1 PROCESS FOR PRODUCING α-(N,N DIALKYL)-AMINO CARBOXYLIC ACID AMIDES BASF AKTIENGESELLSCHAFT (DE) 1997-02-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090036523-A1 PRODRUGS OF CANNABIDIOL, COMPOSITIONS COMPRISING PRODRUGS OF CANNABIDIOL AND METHODS OF USING THE SAME CNR2, CNR1, FAAH ALDH1A1 1490/4885LMNA 1353/4885MEN1 3729/4885
US-20110052694-A1 USE OF CANNABIDIOL PRODRUGS IN TOPICAL AND TRANSDERMAL ADMINISTRATION WITH MICRONEEDLES PNLIP, CNR2, CNR1 ALDH1A1 3684/4885LMNA 3547/4885MEN1 1518/4885
US-11572342-B2 Antimicrobial and antiviral sulfur containing glycerol monoester derivatives MAVS, SARS1, MGLL ALDH1A1 3686/4885LMNA 4761/4885MEN1 3893/4885
US-11873272-B2 Antimicrobial and antiviral sulfur containing glycerol monoester derivatives MAVS, SARS1, MGLL ALDH1A1 3686/4885LMNA 4761/4885MEN1 3893/4885
US-20230174473-A1 ANTIMICROBIAL AND ANTIVIRAL SULFUR CONTAINING GLYCEROL MONOESTER DERIVATIVES MAVS, SARS1, MGLL ALDH1A1 3686/4885LMNA 4761/4885MEN1 3893/4885
US-20150197484-A1 USE OF CANNABIDIOL PRODRUGS IN TOPICAL AND TRANSDERMAL ADMINISTRATION WITH MICRONEEDLES PNLIP, CNR2, CNR1 ALDH1A1 3684/4885LMNA 3547/4885MEN1 1518/4885
US-11365176-B2 Antimicrobial and antiviral sulfur containing glycerol monoester derivatives MAVS, SARS1, MGLL ALDH1A1 3686/4885LMNA 4761/4885MEN1 3893/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.