SCHEMBL14907146

SCHEMBL14907146

CCOC(=O)Cc1nnc(C)o1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.59
CA12 O43570 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA9 Q16790 1/20 0.45
HSD17B10 Q99714 2/20 0.41
PKM P14618 1/20 0.41
ATM Q13315 1/20 0.41
MAPK1 P28482 2/20 0.41
MGAM O43451 1/20 0.40
GAA P10253 1/20 0.40
SI P14410 1/20 0.40
MGAM2 Q2M2H8 1/20 0.40
APLNR P35414 1/20 0.39
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 1/20 0.38
HPGD P15428 1/20 0.38
TRPA1 O75762 1/20 0.38
POLB P06746 1/20 0.37
MEN1 O00255 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12343975 0.85 SMN1; SMN2 (0.59) SMN1; SMN2CA12CA1CA2CA9
SCHEMBL26384544 0.82 SMN1; SMN2 (0.56) SMN1; SMN2CA12CA1CA2CA9
SCHEMBL3822584 0.82 SMN1; SMN2 (0.56) SMN1; SMN2CA12CA1CA2CA9
SCHEMBL11608428 0.82 SMN1; SMN2 (0.56) SMN1; SMN2CA12CA1CA2CA9
SCHEMBL28987822 0.81 SMN1; SMN2 (0.55) SMN1; SMN2CA12CA1CA2CA9
SCHEMBL3823100 0.80 SMN1; SMN2 (0.54) SMN1; SMN2CA12CA1CA2CA9
SCHEMBL20651164 0.80 SMN1; SMN2 (0.54) SMN1; SMN2CA12CA1CA2CA9
SCHEMBL13140041 0.80 SMN1; SMN2 (0.54) SMN1; SMN2CA12CA1CA2CA9
SCHEMBL28987842 0.78 SMN1; SMN2 (0.56) SMN1; SMN2CA12CA1CA2CA9
SCHEMBL26849768 0.78 SMN1; SMN2 (0.56) SMN1; SMN2CA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 37 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026099466-A1 TARGETED PROTEIN DEGRADATION MONTE ROSA THERAPEUTICS AG (CH) 2026-05-15 WO disclosed
US-11851449-B2 Heterocyclic amide compounds having an RORvt inhibitory action TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2023-12-26 US disclosed
EP-3018123-B1 AMIDE COMPOUND TAKEDA PHARMACEUTICALS CO (JP) 2023-05-10 EP disclosed
CN-114835656-A 1,3, 4-oxadiazole ethyl acetate and synthesis method thereof 天津中医药大学 2022-08-02 CN disclosed
US-20210277030-A1 AMIDE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2021-09-09 US disclosed
CN-108473426-B Cyclic amine derivative and medical use thereof 东丽株式会社 2021-09-07 CN disclosed
US-11053262-B2 Heterocyclic amide compounds having RORyT inhibitory action TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2021-07-06 US disclosed
US-10881649-B2 Therapeutic agent or preventive agent for alopecia areata TORAY INDUSTRIES, INC. (JP) 2021-01-05 US disclosed
US-10881649-B2 Therapeutic agent or preventive agent for alopecia areata TORAY INDUSTRIES, INC. (JP) 2021-01-05 US disclosed
EP-3746079-A1 ANTIBODY DRUG CONJUGATES (ADCS) WITH NAMPT INHIBITORS Bayer Aktiengesellschaft (DE) 2020-12-09 EP disclosed
WO-2017131156-A1 CYCLIC AMINE DERIVATIVE AND PHARMACEUTICAL USE THEREOF 東レ株式会社 2017-08-03 WO disclosed
US-20170107240-A1 AMIDE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2017-04-20 US disclosed
US-20170050974-A1 HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2017-02-23 US disclosed
EP-3018123-A1 AMIDE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2016-05-11 EP disclosed
EP-3018126-A1 HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2016-05-11 EP disclosed
US-9221841-B2 Mitotic kinesin inhibitors and methods of use thereof ARRAY BIOPHARMA INC. (US) 2015-12-29 US disclosed
US-20150191490-A1 MITOTIC KINESIN INHIBTORS AND METHODS OF USE THEREOF ARRAY BIOPHARMA INC. (US) 2015-07-09 US disclosed
US-20140018399-A1 MITOTIC KINESIN INHIBTORS AND METHODS OF USE THEREOF ARRAY BIOPHARMA INC. (US) 2014-01-16 US disclosed
US-8580828-B2 Mitotic kinesin inhibitors and methods of use thereof ARRAY BIOPHARMA INC. (US) 2013-11-12 US disclosed
US-20130109656-A1 MITOTIC KINESIN INHIBITORS AND METHODS OF USE THEREOF ARRAY BIOPHARMA, INC. 2013-05-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130109656-A1 MITOTIC KINESIN INHIBITORS AND METHODS OF USE THEREOF KIF5B, KIF2C, KIFC1 SMN1; SMN2 1336/4885CA12 3624/4885CA1 2463/4885
US-20150191490-A1 MITOTIC KINESIN INHIBTORS AND METHODS OF USE THEREOF KIF5B, KIF2C, KIFC1 SMN1; SMN2 1710/4885CA12 2542/4885CA1 1169/4885
US-20170050974-A1 HETEROCYCLIC COMPOUND RORC, RORB, RORA SMN1; SMN2 4127/4885CA12 1747/4885CA1 681/4885
US-20170107240-A1 AMIDE COMPOUND RORB, RORC, RORA SMN1; SMN2 4136/4885CA12 1061/4885CA1 311/4885
US-10881649-B2 Therapeutic agent or preventive agent for alopecia areata RORA, RORB, RORC SMN1; SMN2 4834/4885CA12 647/4885CA1 599/4885
US-20210277030-A1 AMIDE COMPOUND RORB, RORC, RORA SMN1; SMN2 4136/4885CA12 1061/4885CA1 311/4885
US-20140018399-A1 MITOTIC KINESIN INHIBTORS AND METHODS OF USE THEREOF KIF5B, KIF2C, KIFC1 SMN1; SMN2 1710/4885CA12 2542/4885CA1 1169/4885
US-11851449-B2 Heterocyclic amide compounds having an RORvt inhibitory action RORB, RORC, RORA SMN1; SMN2 3917/4885CA12 852/4885CA1 162/4885
US-11053262-B2 Heterocyclic amide compounds having RORyT inhibitory action RORC, RORB, RORA SMN1; SMN2 4241/4885CA12 527/4885CA1 199/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.