SCHEMBL14939140

SCHEMBL14939140

COc1ccc(CN2CCC(C3(c4cccc(C)c4)Cc4ccccc4C3=O)CC2)cc1

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CXCR3 P49682 4/20 0.53
SIGMAR1 Q99720 2/20 0.50
DRD2 P14416 1/20 0.50
HTR2A P28223 1/20 0.50
HTR2C P28335 1/20 0.50
HTR2B P41595 1/20 0.50
CHRM2 P08172 1/20 0.46
CHRM3 P20309 1/20 0.46
ACHE P22303 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14940471 0.91 CXCR3 (0.48) CXCR3SIGMAR1DRD2HTR2AHTR2C
SCHEMBL14940057 0.91 CXCR3 (0.63) CXCR3SIGMAR1DRD2HTR2AHTR2C
SCHEMBL14938853 0.85 CXCR4 (0.48) DRD2CHRM2CHRM3ACHE
SCHEMBL14939344 0.85 CHRM2 (0.52) CXCR3DRD2CHRM2CHRM3ACHE
SCHEMBL14939321 0.84 SIGMAR1 (0.55) CXCR3SIGMAR1DRD2CHRM2CHRM3
SCHEMBL14939041 0.84 HTR7 (0.40) CXCR3CHRM2CHRM3
SCHEMBL14939226 0.83 CXCR3 (0.61) CXCR3SIGMAR1DRD2HTR2AHTR2C
SCHEMBL14939192 0.83 ALDH1A1 (0.49) SIGMAR1DRD2ACHE
SCHEMBL14939665 0.83 ACHE (0.44) CXCR3DRD2CHRM2CHRM3ACHE
SCHEMBL14940366 0.83 ACHE (0.44) CXCR3DRD2CHRM2CHRM3ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO claimed
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed