SCHEMBL14940366

SCHEMBL14940366

Cc1cccc([C@@]2(C3CCN(Cc4ccccc4C)CC3)Cc3ccccc3C2=O)c1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.44
ALDH1A1 P00352 2/20 0.42
PARP1 P09874 1/20 0.40
KMT2A Q03164 1/20 0.40
HTR7 P34969 1/20 0.39
CXCR3 P49682 1/20 0.39
CHRM2 P08172 1/20 0.38
CHRM3 P20309 1/20 0.38
DRD4 P21917 3/20 0.38
DRD2 P14416 1/20 0.38
GAA P10253 1/20 0.37
UBE2M P61081 1/20 0.37
DCUN1D1 Q96GG9 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14939163 1.00 ACHE (0.44) ACHEALDH1A1PARP1KMT2AHTR7
SCHEMBL14939665 1.00 ACHE (0.44) ACHEALDH1A1PARP1KMT2AHTR7
SCHEMBL14939041 0.93 HTR7 (0.40) ALDH1A1PARP1HTR7CXCR3CHRM2
SCHEMBL14940089 0.91 ACHE (0.48) ACHEALDH1A1PARP1KMT2ACXCR3
SCHEMBL14938989 0.90 HTR7 (0.37) ALDH1A1HTR7CXCR3CHRM2CHRM3
SCHEMBL14938853 0.89 CXCR4 (0.48) ACHEALDH1A1KMT2ACHRM2CHRM3
SCHEMBL14940471 0.88 CXCR3 (0.48) ACHECXCR3CHRM2CHRM3DRD2
SCHEMBL14939601 0.88 ALDH1A1 (0.46) ACHEALDH1A1PARP1KMT2ACXCR3
SCHEMBL14939161 0.86 ALDH1A1 (0.39) ALDH1A1HTR7CXCR3CHRM2CHRM3
SCHEMBL14939344 0.84 CHRM2 (0.52) ACHEALDH1A1CXCR3CHRM2CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO claimed
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed