SCHEMBL14939601

SCHEMBL14939601

Cc1cccc(C2(C3CCN(Cc4ccccc4C(F)(F)F)CC3)Cc3ccccc3C2=O)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.46
KDM4E B2RXH2 7/20 0.46
TDP1 Q9NUW8 4/20 0.43
KMT2A Q03164 4/20 0.43
NPSR1 Q6W5P4 3/20 0.43
ATM Q13315 3/20 0.43
MEN1 O00255 3/20 0.43
GAA P10253 2/20 0.43
POLB P06746 1/20 0.43
BCHE P06276 1/20 0.43
ACHE P22303 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
PARP1 P09874 1/20 0.42
RECQL P46063 1/20 0.39
CXCR3 P49682 1/20 0.39
MAPT P10636 1/20 0.38
ALOX15 P16050 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14939041 0.89 HTR7 (0.40) ALDH1A1PARP1CXCR3
SCHEMBL14939665 0.88 ACHE (0.44) ALDH1A1KMT2AGAAACHEPARP1
SCHEMBL14940366 0.88 ACHE (0.44) ALDH1A1KMT2AGAAACHEPARP1
SCHEMBL14939163 0.88 ACHE (0.44) ALDH1A1KMT2AGAAACHEPARP1
SCHEMBL14938989 0.85 HTR7 (0.37) ALDH1A1CXCR3
SCHEMBL14938853 0.85 CXCR4 (0.48) ALDH1A1KMT2AMEN1BCHEACHE
SCHEMBL14940471 0.84 CXCR3 (0.48) NPSR1ACHECXCR3
SCHEMBL14939161 0.84 ALDH1A1 (0.39) ALDH1A1TDP1CXCR3
SCHEMBL14939344 0.80 CHRM2 (0.52) ALDH1A1KDM4EACHECXCR3
SCHEMBL14939140 0.79 CXCR3 (0.53) ACHECXCR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO claimed
WO-2013068785-A1 INDANONE AND INDANDIONE DERIVATIVES AND HETEROCYCLIC ANALOGS ACTELION PHARMACEUTICALS LTD (CH) 2013-05-16 WO disclosed