SCHEMBL14965623

SCHEMBL14965623

O=[N+]([O-])c1cn2c(n1)OCCN(Cc1ccccc1Br)CC2

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP2A13 Q16696 1/20 0.48
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
POLB P06746 3/20 0.40
KDM4E B2RXH2 4/20 0.40
ALDH1A1 P00352 4/20 0.40
LMNA P02545 1/20 0.40
HTR6 P50406 1/20 0.39
FAAH O00519 1/20 0.38
RAB9A P51151 1/20 0.37
CASP1 P29466 1/20 0.36
CASP4 P49662 1/20 0.36
CASP5 P51878 1/20 0.36
ATM Q13315 1/20 0.36
TSHR P16473 1/20 0.36
RECQL P46063 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
ACHE P22303 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14965682 0.85 HTR7 (0.44) MEN1KMT2APOLBKDM4EALDH1A1
SCHEMBL14965773 0.84 L3MBTL1 (0.46) MEN1KMT2APOLBKDM4EALDH1A1
SCHEMBL14965999 0.83 ALDH1A1 (0.43) POLBKDM4EALDH1A1LMNAFAAH
SCHEMBL14965974 0.82 FAAH (0.41) MEN1KMT2APOLBKDM4EALDH1A1
SCHEMBL14965699 0.81 SMN1; SMN2 (0.43) MEN1KMT2APOLBKDM4EALDH1A1
SCHEMBL14971108 0.81 ALDH1A1 (0.44) KDM4EALDH1A1LMNAFAAHRAB9A
SCHEMBL14965813 0.81 ALDH1A1 (0.53) MEN1KMT2APOLBKDM4EALDH1A1
SCHEMBL14965655 0.80 PDE4B (0.36) MEN1KMT2APOLBALDH1A1CASP1
SCHEMBL14965939 0.80 PDE9A (0.39) MEN1KMT2APOLBKDM4EALDH1A1
SCHEMBL14966128 0.79 ALDH1A1 (0.38) ALDH1A1LMNAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed