SCHEMBL14965726

SCHEMBL14965726

Cc1ccc(NC(=O)N2CCOc3nc([N+](=O)[O-])cn3CC2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
TP53 P04637 3/20 0.43
KDM4E B2RXH2 2/20 0.43
ALDH1A1 P00352 2/20 0.43
GAA P10253 4/20 0.42
MAPT P10636 4/20 0.42
TSHR P16473 1/20 0.41
KMT2A Q03164 2/20 0.40
HTT P42858 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
FAAH O00519 2/20 0.40
POLB P06746 2/20 0.40
MEN1 O00255 1/20 0.39
ESR2 Q92731 1/20 0.39
BLM P54132 1/20 0.39
LMNA P02545 1/20 0.39
ABL1 P00519 1/20 0.39
RIN1 Q13671 1/20 0.39
TDP1 Q9NUW8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14966280 0.90 SMN1; SMN2 (0.52) NPC1RAB9AALDH1A1GAAMAPT
SCHEMBL14965955 0.90 MAPK1 (0.44) KDM4EALDH1A1GAAMAPTSMN1; SMN2
SCHEMBL14965945 0.89 BLM (0.55) ALDH1A1MAPTTSHRKMT2AHTT
SCHEMBL14965906 0.87 PANK3 (0.42) GAAMAPTHTTSMN1; SMN2FAAH
SCHEMBL14965486 0.85 LMNA (0.42) TP53KDM4EALDH1A1GAAMAPT
SCHEMBL14966116 0.78 MAPT (0.46) NPC1RAB9AKDM4EALDH1A1MAPT
SCHEMBL14965869 0.77 ALDH1A1 (0.41) NPC1ALDH1A1GAAMAPTKMT2A
SCHEMBL14966075 0.77 KDM4E (0.46) TP53KDM4EALDH1A1KMT2AHTT
SCHEMBL14965880 0.76 P2RY12 (0.38) KDM4EALDH1A1KMT2APOLBLMNA
SCHEMBL14965783 0.76 NPC1 (0.51) NPC1KDM4EALDH1A1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed