SCHEMBL14965864

SCHEMBL14965864

O=C(O)CN1CCC(N2CCOc3nc([N+](=O)[O-])cn3CC2)CC1

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.39
ITGA2B P08514 1/20 0.39
ALOX15 P16050 1/20 0.38
CHRM1 P11229 1/20 0.33
KDM4E B2RXH2 2/20 0.33
ALDH1A1 P00352 1/20 0.33
KMT2A Q03164 1/20 0.32
KCNH2 Q12809 3/20 0.31
LMNA P02545 1/20 0.31
ACHE P22303 1/20 0.30
USP5 P45974 1/20 0.30
TRPV6 Q9H1D0 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14965582 0.87 HSD17B10 (0.38) CHRM1ALDH1A1KMT2AKCNH2LMNA
SCHEMBL14966094 0.82 PDE7A (0.33) CHRM1
SCHEMBL14965938 0.81 CHRM1 (0.34) CHRM1KMT2AKCNH2
SCHEMBL14965838 0.81 CHRM1 (0.34) CHRM1KMT2AKCNH2
SCHEMBL14965829 0.79 ALDH1A1 (0.39) KDM4EALDH1A1LMNA
SCHEMBL14965756 0.76 PKM (0.40) KDM4EALDH1A1LMNA
SCHEMBL14965802 0.76 L3MBTL3 (0.43) KMT2ALMNA
SCHEMBL14966168 0.75 ALDH1A1 (0.40) KDM4EALDH1A1KMT2ALMNA
SCHEMBL14965832 0.75 NPC1 (0.36) ALOX15CHRM1ALDH1A1KMT2ALMNA
SCHEMBL14965791 0.74 KDM4E (0.36) CHRM1KDM4EALDH1A1KMT2AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed