SCHEMBL14965802

SCHEMBL14965802

O=C(c1ccc(C(F)(F)F)cc1)N1CCC(N2CCOc3nc([N+](=O)[O-])cn3CC2)CC1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
L3MBTL3 Q96JM7 9/20 0.43
L3MBTL1 Q9Y468 7/20 0.43
GAA P10253 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
HPGD P15428 2/20 0.41
LMNA P02545 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
SCN9A Q15858 1/20 0.41
SCN10A Q9Y5Y9 1/20 0.41
HSD11B1 P28845 2/20 0.40
MBTD1 Q05BQ5 4/20 0.40
TP53BP1 Q12888 1/20 0.40
L3MBTL4 Q8NA19 1/20 0.40
MGLL Q99685 2/20 0.40
MEN1 O00255 1/20 0.39
TSHR P16473 1/20 0.39
KMT2A Q03164 1/20 0.39
SLC2A1 P11166 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14965688 0.90 RBP4 (0.45) L3MBTL3L3MBTL1GAATDP1HPGD
SCHEMBL14965608 0.89 CHRM1 (0.48) L3MBTL3L3MBTL1SCN9AHSD11B1MBTD1
SCHEMBL14965829 0.78 ALDH1A1 (0.39) LMNA
SCHEMBL14965709 0.77 CHRM1 (0.46) SCN9A
SCHEMBL14965755 0.77 EPHX2 (0.50)
SCHEMBL14965651 0.76 HPGD (0.43) GAAHPGDLMNATSHRKMT2A
SCHEMBL14965864 0.76 ITGB3 (0.39) LMNAKMT2A
SCHEMBL14965843 0.75 CHRM1 (0.48) HPGDLMNASMN1; SMN2HSD11B1MGLL
SCHEMBL14965838 0.75 CHRM1 (0.34) MEN1KMT2A
SCHEMBL14965938 0.75 CHRM1 (0.34) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed