SCHEMBL14965973

SCHEMBL14965973

O=C(Cc1ccc(OC(F)(F)F)cc1)NC1CCC(N2CCOc3nc([N+](=O)[O-])cn3CC2)CC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 1/20 0.51
KCNH2 Q12809 4/20 0.44
EPHX2 P34913 3/20 0.43
PTGS1 P23219 1/20 0.40
SLC6A2 P23975 1/20 0.40
SLC6A4 P31645 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.38
TMEM97 Q5BJF2 1/20 0.37
MCHR1 Q99705 2/20 0.36
MMP1 P03956 1/20 0.36
MMP3 P08254 1/20 0.36
MMP7 P09237 1/20 0.36
MMP9 P14780 1/20 0.36
MMP8 P22894 1/20 0.36
MMP13 P45452 1/20 0.36
MMP14 P50281 1/20 0.36
CCNA2 P20248 1/20 0.35
CDK2 P24941 1/20 0.35
CCNA1 P78396 1/20 0.35
SIGMAR1 Q99720 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14965709 0.89 CHRM1 (0.46) CHRM1KCNH2EPHX2PTGS1SLC6A2
SCHEMBL14965728 0.88 EPHX2 (0.47) CHRM1EPHX2FAAH
SCHEMBL14965836 0.83 MCHR1 (0.41) CHRM1KCNH2EPHX2PTGS1SLC6A2
SCHEMBL14965608 0.82 CHRM1 (0.48) CHRM1KCNH2EPHX2PTGS1SLC6A2
SCHEMBL14965755 0.81 EPHX2 (0.50) CHRM1KCNH2EPHX2PTGS1SLC6A2
SCHEMBL14966094 0.80 PDE7A (0.33) CHRM1SIGMAR1
SCHEMBL14971162 0.78 DRD2 (0.38) CHRM1
SCHEMBL14965548 0.77 CHRM1 (0.52) CHRM1KCNH2PTGS1SLC6A2SLC6A4
SCHEMBL14965842 0.76 CHRM1 (0.59) CHRM1KCNH2PTGS1SLC6A2SLC6A4
SCHEMBL14965622 0.75 CHRM1 (0.50) CHRM1KCNH2PTGS1SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed