SCHEMBL14965709

SCHEMBL14965709

O=C(NC1CCC(N2CCOc3nc([N+](=O)[O-])cn3CC2)CC1)c1ccc(OC(F)(F)F)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 1/20 0.46
KCNH2 Q12809 6/20 0.44
MCHR1 Q99705 1/20 0.40
DPP4 P27487 1/20 0.40
DPP8 Q6V1X1 1/20 0.40
DPP9 Q86TI2 1/20 0.40
DPP7 Q9UHL4 1/20 0.40
PTGS1 P23219 1/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
IDH1 O75874 3/20 0.37
SCN5A Q14524 2/20 0.37
SCN9A Q15858 2/20 0.37
SLC6A5 Q9Y345 1/20 0.37
HPGDS O60760 1/20 0.36
HDAC4 P56524 1/20 0.36
FAAH O00519 2/20 0.35
EPHX2 P34913 2/20 0.35
RAF1 P04049 1/20 0.35
LIPE Q05469 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14965836 0.91 MCHR1 (0.41) CHRM1KCNH2MCHR1PTGS1SLC6A2
SCHEMBL14965973 0.89 CHRM1 (0.51) CHRM1KCNH2MCHR1PTGS1SLC6A2
SCHEMBL14965728 0.89 EPHX2 (0.47) CHRM1FAAHEPHX2
SCHEMBL14965608 0.86 CHRM1 (0.48) CHRM1KCNH2PTGS1SLC6A2SLC6A4
SCHEMBL14965755 0.82 EPHX2 (0.50) CHRM1KCNH2MCHR1PTGS1SLC6A2
SCHEMBL14966094 0.81 PDE7A (0.33) CHRM1
SCHEMBL30260105 0.81 CHRM1 (0.61) CHRM1KCNH2MCHR1DPP4DPP8
SCHEMBL14971162 0.79 DRD2 (0.38) CHRM1
SCHEMBL14965365 0.77 CHRM1 (0.49) CHRM1KCNH2PTGS1SLC6A2SLC6A4
SCHEMBL14965802 0.77 L3MBTL3 (0.43) SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed