SCHEMBL14965836

SCHEMBL14965836

O=C(NC1CCC(N2CCOc3nc([N+](=O)[O-])cn3CC2)CC1)c1cccc(OC(F)(F)F)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 1/20 0.41
CHRM1 P11229 1/20 0.41
TAS1R3 Q7RTX0 1/20 0.40
TAS1R1 Q7RTX1 1/20 0.40
TAS1R2 Q8TE23 1/20 0.40
KCNH2 Q12809 4/20 0.38
PDE4B Q07343 1/20 0.38
PDE4D Q08499 1/20 0.38
ALDH1A1 P00352 1/20 0.38
NPC1 O15118 1/20 0.37
ROCK2 O75116 1/20 0.36
HPGDS O60760 2/20 0.36
EPHX2 P34913 1/20 0.36
CCR2 P41597 2/20 0.36
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
TMEM97 Q5BJF2 1/20 0.35
PTGS1 P23219 1/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14965709 0.91 CHRM1 (0.46) MCHR1CHRM1KCNH2HPGDSEPHX2
SCHEMBL14965728 0.83 EPHX2 (0.47) CHRM1EPHX2
SCHEMBL14965973 0.83 CHRM1 (0.51) MCHR1CHRM1KCNH2EPHX2TMEM97
SCHEMBL14965608 0.79 CHRM1 (0.48) CHRM1KCNH2EPHX2PTGS1SLC6A2
SCHEMBL14966094 0.79 PDE7A (0.33) CHRM1
SCHEMBL14965916 0.77 ABL1 (0.56) MCHR1CHRM1KCNH2ALDH1A1NPC1
SCHEMBL14965755 0.77 EPHX2 (0.50) MCHR1CHRM1KCNH2EPHX2PTGS1
SCHEMBL14971162 0.77 DRD2 (0.38) CHRM1
SCHEMBL14966212 0.76 HSD11B1 (0.44) CHRM1KCNH2ALDH1A1
SCHEMBL14965621 0.75 CHRM1 (0.44) CHRM1KCNH2ALDH1A1PTGS1SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO claimed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed
WO-2013072903-A1 NITROIMIDAZOXADIAZOCINE COMPOUNDS ITHEMBA PHARMACEUTICALS (PROPRIETARY) LIMITED (ZA) 2013-05-23 WO disclosed